SCHEMBL6161235

SCHEMBL6161235

CC(C)CC(NC(=O)COc1ccc(CCOc2ccccc2C(=O)O)cc1)c1ccc(C(F)(F)F)cc1

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ABCC8 Q09428 2/20 0.43
CCR5 P51681 1/20 0.41
ENPP2 Q13822 1/20 0.41
SIRT2 Q8IXJ6 1/20 0.40
PSMB5 P28074 2/20 0.40
ADAMTS5 Q9UNA0 1/20 0.40
HCAR2 Q8TDS4 1/20 0.40
SLC22A1 O15245 1/20 0.40
ABCC3 O15438 1/20 0.40
ABCC4 O15439 1/20 0.40
NR1I2 O75469 1/20 0.40
ABCB11 O95342 1/20 0.40
LMNA P02545 1/20 0.40
CYP3A4 P08684 1/20 0.40
ADORA3 P0DMS8 1/20 0.40
HTR2A P28223 1/20 0.40
MAPK1 P28482 1/20 0.40
ADRA1A P35348 1/20 0.40
PTGS2 P35354 1/20 0.40
PDE4D Q08499 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6160652 0.83 ENPP2 (0.41) ENPP2SIRT2PSMB5PPARAPPARD
SCHEMBL3996205 0.79 PSMB5 (0.43) ENPP2SIRT2PSMB5PPARAPPARD
SCHEMBL6160660 0.78 ENPP2 (0.42) ENPP2SIRT2PSMB5PPARAPPARD
SCHEMBL6160047 0.77 SIRT2 (0.39) SIRT2PSMB5LMNAPPARAPPARD
SCHEMBL4962776 0.74 TRPM8 (0.54) PSMB5LMNAMAPK1PPARAPPARD
SCHEMBL3996571 0.73 PSMB5 (0.43) SIRT2PSMB5PPARAPPARD
SCHEMBL6160055 0.72 SIRT2 (0.41) ENPP2SIRT2PSMB5LMNAPPARA
SCHEMBL6161238 0.72 SLC2A1 (0.44) SIRT2PPARAPPARD
SCHEMBL6160658 0.71 SIRT2 (0.43) ENPP2SIRT2PPARAPPARD
SCHEMBL2448991 0.68 ALDH1A1 (0.59) HCAR2LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1517680-A1 BENZOIC ACID DERIVATIVES AS MODULATORS OF PPAR ALPHA AND GAMMA Astrazeneca AB (SE) 2005-03-30 EP claimed
WO-2004000295-A1 BENZOIC ACID DERIVATIVES AS MODULATORS OF PPAR ALPHA AND GAMMA ASTRAZENECA AB (SE) 2003-12-31 WO claimed