SCHEMBL6166963

SCHEMBL6166963

O=C(O)c1cccc(-c2cocn2)c1

nearest known ligand 0.55

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
KMO O15229 2/20 0.53
SCN9A Q15858 2/20 0.49
KEAP1 Q14145 1/20 0.49
RXRA P19793 2/20 0.47
RXRB P28702 2/20 0.47
DDT P30046 1/20 0.47
CD74 P04233 1/20 0.46
MIF P14174 1/20 0.46
L3MBTL1 Q9Y468 2/20 0.44
KDM4E B2RXH2 1/20 0.44
ALDH1A1 P00352 1/20 0.44
POLB P06746 1/20 0.44
TDP1 Q9NUW8 1/20 0.44
HDAC4 P56524 1/20 0.44
NPC1 O15118 1/20 0.43
RAB9A P51151 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3840412 0.86 SCN9A (0.49) KMOSCN9AHDAC4
SCHEMBL6163665 0.81 GABRG2 (0.51) SCN9AKDM4ENPC1RAB9A
SCHEMBL4765377 0.81 HDAC4 (0.50) KDM4EALDH1A1POLBHDAC4NPC1
SCHEMBL14564377 0.79 SCN9A (0.62) KMOSCN9AHDAC4
SCHEMBL4751198 0.77 HSD17B1 (0.58) SCN9A
SCHEMBL2986666 0.76 DHODH (0.50) RXRARXRBKDM4EALDH1A1POLB
SCHEMBL648786 0.76 SCN9A (0.53) SCN9AMIFTDP1HDAC4NPC1
SCHEMBL29904709 0.75 KMO (0.86) KMOKEAP1RXRARXRBCD74
SCHEMBL71238 0.75 KMO (0.86) KMOKEAP1RXRARXRBCD74
SCHEMBL30725957 0.75 KMO (0.86) KMOKEAP1RXRARXRBCD74

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1379511-B1 DIHYDRO-BENZO (b) (1, 4) DIAZEPIN-2-ONE DERIVATIVES AS MGLUR2 ANTAGONISTS II HOFFMANN LA ROCHE (CH) 2005-07-20 EP disclosed