SCHEMBL6172246

SCHEMBL6172246

COc1ccc2[nH]c(C(=O)c3cccc(C)c3)c(C(C(=O)O)C(=O)O)c2c1

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 8/20 0.45
MEN1 O00255 7/20 0.45
MAPT P10636 4/20 0.45
GAA P10253 4/20 0.45
PTGS1 P23219 1/20 0.45
PTGS2 P35354 1/20 0.45
KDM4E B2RXH2 5/20 0.44
ALDH1A1 P00352 5/20 0.44
HPGD P15428 3/20 0.44
NPC1 O15118 1/20 0.44
RAB9A P51151 1/20 0.44
HSD17B10 Q99714 3/20 0.43
TUBB4A P04350 3/20 0.43
TUBB P07437 3/20 0.43
TUBA3C P0DPH7 3/20 0.43
TUBA1B P68363 3/20 0.43
TUBA4A P68366 3/20 0.43
TUBB4B P68371 3/20 0.43
TUBB3 Q13509 3/20 0.43
TUBB2A Q13885 3/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7203928 0.89 ALDH1A1 (0.52) KMT2AMEN1MAPTGAAPTGS1
SCHEMBL6170675 0.84 MAP2 (0.44) KMT2AMEN1MAPTPTGS1PTGS2
SCHEMBL6168282 0.80 PTGS2 (0.68) KMT2AMEN1MAPTGAAPTGS1
SCHEMBL27569322 0.80 KMT2A (0.46) KMT2AMEN1MAPTGAAPTGS1
SCHEMBL8140742 0.79 MEN1 (0.48) KMT2AMEN1MAPTGAAPTGS1
SCHEMBL8140740 0.78 MEN1 (0.49) KMT2AMEN1MAPTGAAPTGS1
SCHEMBL6170113 0.78 ENPP2 (0.43) KMT2AMEN1MAPTPTGS1PTGS2
SCHEMBL6170210 0.75 MAP2 (0.46) KMT2AMEN1MAPTPTGS1PTGS2
SCHEMBL7206101 0.74 ALDH1A1 (0.48) KMT2AMEN1MAPTGAAPTGS2
SCHEMBL6172849 0.74 ALDH1A1 (0.42) KMT2AMEN1MAPTGAAPTGS1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1045833-B1 2,3-SUBSTITUTED INDOLE COMPOUNDS AS COX-2 INHIBITORS PFIZER (US) 2005-11-02 EP disclosed