SCHEMBL6204079

SCHEMBL6204079

COCO[CH]c1cc(F)cc(F)c1

nearest known ligand 0.40

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
PTGS1 P23219 1/20 0.34
PTGS2 P35354 1/20 0.34
NFE2L2 Q16236 2/20 0.31
IDO1 P14902 1/20 0.30
RELA Q04206 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6204739 0.81 NFE2L2 (0.49) PTGS1PTGS2NFE2L2RELA
SCHEMBL6205425 0.79 NFE2L2 (0.44) PTGS1NFE2L2
SCHEMBL16961847 0.75 PTGS1 (0.40) PTGS1PTGS2NFE2L2IDO1RELA
SCHEMBL27624827 0.71 TRPA1 (0.41)
SCHEMBL5410674 0.70 TRPA1 (0.39) NFE2L2IDO1RELA
SCHEMBL8140047 0.67 SOD1 (0.40) IDO1
SCHEMBL6203320 0.66 RELA (0.47) NFE2L2IDO1RELA
SCHEMBL6203560 0.66 ALDH1A1 (0.46) IDO1
Methoxymethane SCHEMBL27837378 0.65 CA12 (0.47) PTGS1PTGS2NFE2L2IDO1
SCHEMBL7563502 0.64 NFE2L2 (0.47) PTGS1PTGS2NFE2L2RELA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1506175-A1 N-SUBSTITUTED TRICYCLIC 3-AMINOPYRAZOLES AS PDGF RECEPTOR INHIBITORS JANSSEN PHARMACEUTICA N.V. (BE) 2005-02-16 EP disclosed
WO-2003097609-A1 N-SUBSTITUTED TRICYCLIC 3-AMINOPYRAZOLES AS PDFG RECEPTOR INHIBITORS JANSSEN PHARMACEUTICA N.V. (BE) 2003-11-27 WO disclosed