SCHEMBL6231994

SCHEMBL6231994

Nc1ccc2sc(CN3CCCCC3)cc2c1

nearest known ligand 0.47

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.47
DRD2 P14416 2/20 0.47
MAOA P21397 1/20 0.47
ACHE P22303 2/20 0.45
MCHR1 Q99705 2/20 0.43
ADORA2A P29274 8/20 0.42
ADORA1 P30542 7/20 0.42
KDM4E B2RXH2 1/20 0.39
MAPT P10636 1/20 0.39
HTT P42858 1/20 0.39
TDP1 Q9NUW8 1/20 0.39
L3MBTL1 Q9Y468 1/20 0.39
DRD4 P21917 1/20 0.39
DRD3 P35462 1/20 0.39
FAAH O00519 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6607240 0.98 DRD2 (0.48) ALDH1A1DRD2MAOAACHEMCHR1
SCHEMBL6235676 0.87 CA2 (0.50) MCHR1ADORA2AADORA1KDM4EMAPT
SCHEMBL6231136 0.85 LMNA (0.50) DRD2MAOAMCHR1KDM4EMAPT
SCHEMBL6251149 0.81 DRD4 (0.50) ALDH1A1DRD2MCHR1KDM4EMAPT
SCHEMBL10238584 0.80 FAAH (0.56) DRD2DRD4DRD3FAAH
SCHEMBL6232410 0.79 MCHR1 (0.49) ALDH1A1DRD2MCHR1KDM4EHTT
SCHEMBL6607124 0.74 ALDH1A1 (0.56) ALDH1A1KDM4EMAPTHTTTDP1
SCHEMBL24601455 0.72 CYP2A6 (0.58) ALDH1A1KDM4EMAPTTDP1
SCHEMBL23612352 0.72 BACE1 (0.41) ALDH1A1KDM4EMAPTTDP1
SCHEMBL2924832 0.71 ALDH1A1 (0.68) ALDH1A1DRD2MAOAACHEKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2004092181-A9 HETEROCYCLIC MCHR1 ANTAGONISTS SMITHKLINE BEECHAM CORP (US) 2005-01-27 WO disclosed