SCHEMBL6236

SCHEMBL6236

C=CCCCN(C)c1c(C)noc1-c1ccc(-c2ccc(C3(CC(=O)OCC)CC3)cc2)cc1

nearest known ligand 0.34

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
GAA P10253 1/20 0.34
BRD4 O60885 2/20 0.33
ABCC3 O15438 1/20 0.31
ABCC4 O15439 1/20 0.31
ABCB11 O95342 1/20 0.31
CYP2C8 P10632 1/20 0.31
CYP2C9 P11712 1/20 0.31
ABCB4 P21439 1/20 0.31
LPAR1 Q92633 1/20 0.31
ABCC2 Q92887 1/20 0.31
SLCO1B3 Q9NPD5 1/20 0.31
SLCO1B1 Q9Y6L6 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6916 0.89 BRD4 (0.33) BRD4ABCC3ABCC4ABCB11CYP2C8
SCHEMBL7501 0.87 ABCC3 (0.37) ABCC3ABCC4ABCB11CYP2C8CYP2C9
SCHEMBL6445 0.85 CHRM1 (0.36) GAA
SCHEMBL6153 0.83 GAA (0.36) GAABRD4ABCC3ABCC4ABCB11
SCHEMBL7532 0.83 ALOX5 (0.35) GAABRD4CYP2C9
SCHEMBL6705 0.82 LPAR1 (0.44) BRD4ABCC3ABCC4ABCB11CYP2C8
SCHEMBL7572 0.81 SLC26A6 (0.36) GAABRD4LPAR1
SCHEMBL6765 0.81 BRD4 (0.33) GAABRD4
SCHEMBL6973 0.81 BRD4 (0.36) GAABRD4CYP2C9
SCHEMBL7632 0.81 KMT2A (0.38) GAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2483252-A2 COMPOUNDS AS LYSOPHOSPHATIDIC ACID RECEPTOR ANTAGONISTS Amira Pharmaceuticals, Inc. (US) 2012-08-08 EP disclosed
WO-2011041694-A2 COMPOUNDS AS LYSOPHOSPHATIDIC ACID RECEPTOR ANTAGONISTS AMIRA PHARMACEUTICALS, INC. (US) 2011-04-07 WO disclosed