SCHEMBL6153

SCHEMBL6153

CCOC(=O)CC1(c2ccc(-c3ccc(-c4onc(C)c4N(C)CCCc4ccccc4Cl)cc3)cc2)CC1

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GAA P10253 2/20 0.36
SLC26A6 Q9BXS9 2/20 0.35
RAB9A P51151 1/20 0.34
BRD4 O60885 1/20 0.33
ALDH1A1 P00352 3/20 0.33
ALOX5 P09917 2/20 0.33
ALOX5AP P20292 2/20 0.33
NLRP3 Q96P20 1/20 0.33
CYP4F2 P78329 1/20 0.32
CYP4A11 Q02928 1/20 0.32
LPAR1 Q92633 2/20 0.32
ABCC3 O15438 1/20 0.32
ABCC4 O15439 1/20 0.32
ABCB11 O95342 1/20 0.32
CYP2C8 P10632 1/20 0.32
CYP2C9 P11712 1/20 0.32
ABCB4 P21439 1/20 0.32
ABCC2 Q92887 1/20 0.32
SLCO1B3 Q9NPD5 1/20 0.32
SLCO1B1 Q9Y6L6 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7234 0.90 LPAR1 (0.34) BRD4ALDH1A1ALOX5ALOX5APLPAR1
SCHEMBL7632 0.89 KMT2A (0.38) GAAALDH1A1MAPTP2RX7
SCHEMBL6445 0.89 CHRM1 (0.36) GAASLC26A6RAB9AALDH1A1ALOX5
SCHEMBL1559 0.88 RAB9A (0.39) GAARAB9AALDH1A1LPAR1ABCC3
SCHEMBL6765 0.87 BRD4 (0.33) GAASLC26A6BRD4ALDH1A1ALOX5
SCHEMBL7532 0.84 ALOX5 (0.35) GAABRD4ALDH1A1ALOX5CYP2C9
SCHEMBL7572 0.83 SLC26A6 (0.36) GAASLC26A6BRD4ALDH1A1ALOX5
SCHEMBL6236 0.83 GAA (0.34) GAABRD4LPAR1ABCC3ABCC4
SCHEMBL2214 0.83 LPAR1 (0.45) ALDH1A1ALOX5ALOX5APLPAR1ABCC3
SCHEMBL11897090 0.82 HDAC1 (0.36) RAB9AALDH1A1CYP2C9MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2483252-B1 COMPOUNDS AS LYSOPHOSPHATIDIC ACID RECEPTOR ANTAGONISTS AMIRA PHARMACEUTICALS INC (US) 2017-03-08 EP disclosed
EP-2483252-A2 COMPOUNDS AS LYSOPHOSPHATIDIC ACID RECEPTOR ANTAGONISTS Amira Pharmaceuticals, Inc. (US) 2012-08-08 EP disclosed
WO-2011041694-A2 COMPOUNDS AS LYSOPHOSPHATIDIC ACID RECEPTOR ANTAGONISTS AMIRA PHARMACEUTICALS, INC. (US) 2011-04-07 WO disclosed