SCHEMBL6238840

SCHEMBL6238840

Nc1nc(-c2cccc(C(F)(F)F)c2)co1

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
XDH P47989 1/20 0.52
CTSS P25774 1/20 0.49
IDO1 P14902 1/20 0.48
NOTUM Q6P988 1/20 0.48
ADORA2A P29274 2/20 0.47
ADORA1 P30542 2/20 0.47
BRD4 O60885 1/20 0.47
ATR Q13535 1/20 0.46
KDM1A O60341 2/20 0.46
RAB9A P51151 2/20 0.46
NPC1 O15118 1/20 0.46
TLR8 Q9NR97 1/20 0.45
KMO O15229 1/20 0.45
MAPK1 P28482 2/20 0.44
TSHR P16473 1/20 0.44
PIK3CD O00329 1/20 0.44
PIK3CA P42336 1/20 0.44
PIK3CG P48736 1/20 0.44
GAA P10253 1/20 0.44
KDM4E B2RXH2 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2901258 0.82 LTA4H (0.53) ADORA2AKDM1ATLR8KDM4EIKBKB
SCHEMBL6238252 0.78 LTA4H (0.37) XDHADORA2AADORA1PIK3CAKDM4E
SCHEMBL14564374 0.77 ENPP3 (0.45) ADORA2AADORA1RAB9ANPC1KMO
SCHEMBL6256565 0.76 CTSS (0.60) XDHCTSSIDO1ADORA2AADORA1
SCHEMBL4539598 0.76 RAB9A (0.54) IDO1ADORA2AADORA1RAB9ANPC1
SCHEMBL6234051 0.74 ALOX5AP (0.43) PIK3CAKDM4EALDH1A1
SCHEMBL8110983 0.74 MPL (0.58) IDO1KDM1A
SCHEMBL8119166 0.74 LTA4H (0.54) NOTUMADORA2AADORA1RAB9ANPC1
SCHEMBL1358158 0.73 XDH (0.57) XDHCTSSIDO1ADORA2AADORA1
SCHEMBL474410 0.73 LTA4H (0.67) XDHCTSSRAB9ANPC1KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2005005382-A2 COMPOUNDS, COMPOSITIONS AND METHODS CYTOKINETICS, INC. (US) 2005-01-20 WO disclosed