SCHEMBL628100

SCHEMBL628100

CCOC(=O)C1CCCN(c2nn3cc(I)nc3s2)C1

nearest known ligand 0.54

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
MAPT P10636 17/20 0.54
THRB P10828 2/20 0.54
POLB P06746 2/20 0.50
LMNA P02545 4/20 0.49
TP53 P04637 2/20 0.49
ALDH1A1 P00352 2/20 0.48
SMN1; SMN2 Q16637 1/20 0.48
KDM4E B2RXH2 2/20 0.48
NPSR1 Q6W5P4 2/20 0.48
TSHR P16473 1/20 0.48
CASP1 P29466 1/20 0.48
MMP13 P45452 1/20 0.48
CASP7 P55210 1/20 0.48
GAA P10253 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL628099 0.80 ALDH1A1 (0.49) MAPTTHRBPOLBLMNATP53
SCHEMBL623999 0.77 MAPT (0.55) MAPTTHRBPOLBLMNATP53
SCHEMBL624634 0.77 MAPT (0.52) MAPTTHRBPOLBLMNATP53
SCHEMBL627055 0.76 MAPT (0.48) MAPTTHRBLMNASMN1; SMN2KDM4E
SCHEMBL2561682 0.73 RAB9A (0.67) MAPTTHRBLMNATP53ALDH1A1
SCHEMBL628264 0.73 BTK (0.51) MAPTTHRBPOLB
SCHEMBL30277649 0.72 ALDH1A1 (0.55) MAPTTHRBPOLBLMNATP53
SCHEMBL22061402 0.72 ALDH1A1 (0.55) MAPTTHRBPOLBLMNATP53
SCHEMBL628000 0.71 MAPT (0.42) MAPTTHRBPOLBLMNAGAA
SCHEMBL2565666 0.71 MAPT (0.61) MAPTTHRBTP53ALDH1A1SMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012020217-A1 AMINO- IMIDAZOLOTHIADIAZOLES FOR USE AS PROTEIN OR LIPID KINASE INHIBITORS CENTRO NACIONAL DE INVESTIGACIONES ONCOLÓGICAS (CNIO) (ES) 2012-02-16 WO disclosed
WO-2012020215-A1 AMINO- IMIDAZOLOTHIADIAZOLES FOR USE AS PROTEIN OR LIPID KINASE INHIBITORS CENTRO NACIONAL DE INVESTIGACIONES ONCOLÓGICAS (CNIO) (ES) 2012-02-16 WO disclosed