SCHEMBL627407

SCHEMBL627407

CS(=O)(=O)N1CC2(CCCN(c3nn4cc(I)nc4s3)C2)C1

nearest known ligand 0.41

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
CYP2D6 P10635 8/20 0.41
CYP1A2 P05177 7/20 0.41
ALOX15 P16050 1/20 0.41
ALDH1A1 P00352 7/20 0.41
CYP2C19 P33261 7/20 0.41
HSD17B10 Q99714 5/20 0.41
CYP2C9 P11712 5/20 0.41
MAPK1 P28482 1/20 0.41
CYP3A4 P08684 11/20 0.40
USP2 O75604 3/20 0.39
HPGD P15428 4/20 0.39
TSHR P16473 4/20 0.39
EIF2AK4 Q9P2K8 2/20 0.38
RECQL P46063 1/20 0.35
HIF1A Q16665 2/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL627406 0.80 CYP1A2 (0.46) CYP2D6CYP1A2ALOX15ALDH1A1CYP2C19
SCHEMBL627422 0.78 RET (0.42) CYP2D6CYP1A2ALOX15ALDH1A1CYP2C19
SCHEMBL625703 0.76 MAP3K12 (0.44) EIF2AK4
SCHEMBL627267 0.72 CYP11B2 (0.41) CYP2C19HSD17B10CYP3A4USP2
SCHEMBL627088 0.70 MAPT (0.32)
SCHEMBL628407 0.68 CYP11B2 (0.44) CYP3A4HIF1A
SCHEMBL624035 0.67 SMN1; SMN2 (0.40) ALOX15ALDH1A1HSD17B10USP2HPGD
SCHEMBL625702 0.66 PIK3CA (0.50) CYP2D6CYP1A2ALOX15EIF2AK4
SCHEMBL627168 0.65 CCNE1 (0.39)
SCHEMBL624133 0.65 RORC (0.34) CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012020215-A1 AMINO- IMIDAZOLOTHIADIAZOLES FOR USE AS PROTEIN OR LIPID KINASE INHIBITORS CENTRO NACIONAL DE INVESTIGACIONES ONCOLÓGICAS (CNIO) (ES) 2012-02-16 WO disclosed