SCHEMBL6285244

SCHEMBL6285244

CCCCC(C(=O)Cl)N1C(=O)c2ccccc2C1=O

nearest known ligand 0.55

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 5/20 0.50
POLB P06746 4/20 0.50
KDM4E B2RXH2 1/20 0.50
TP53 P04637 1/20 0.50
GLA P06280 1/20 0.50
CYP3A4 P08684 1/20 0.50
CYP2D6 P10635 1/20 0.50
HPGD P15428 1/20 0.50
ALOX12 P18054 1/20 0.50
NFKB1 P19838 1/20 0.50
APEX1 P27695 1/20 0.50
MAPK1 P28482 1/20 0.50
HSD17B10 Q99714 1/20 0.50
GAA P10253 2/20 0.48
L3MBTL1 Q9Y468 1/20 0.46
ASAH1 Q13510 1/20 0.43
LMNA P02545 1/20 0.42
KMT2A Q03164 1/20 0.41
AADAT Q8N5Z0 1/20 0.40
HIF1A Q16665 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL133528 0.86 POLB (0.68) ALDH1A1POLBKDM4ETP53GLA
SCHEMBL29783279 0.86 POLB (0.68) ALDH1A1POLBKDM4ETP53GLA
SCHEMBL19286640 0.85 ALDH1A1 (0.50) ALDH1A1POLBKDM4ETP53GLA
Hydrochloric Acid SCHEMBL8187825 0.85 POLB (0.66) ALDH1A1POLBKDM4ETP53GLA
Hydrochloric Acid SCHEMBL7757351 0.85 POLB (0.66) ALDH1A1POLBKDM4ETP53GLA
SCHEMBL6243248 0.84 ALDH1A1 (0.53) ALDH1A1POLBKDM4ETP53GLA
SCHEMBL32691108 0.84 ALDH1A1 (0.53) ALDH1A1POLBKDM4ETP53GLA
SCHEMBL29459236 0.84 ALDH1A1 (0.53) ALDH1A1POLBKDM4ETP53GLA
SCHEMBL3195963 0.82 ALDH1A1 (0.48) ALDH1A1POLBKDM4ETP53GLA
SCHEMBL29453019 0.82 ALDH1A1 (0.48) ALDH1A1POLBKDM4ETP53GLA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 8 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8252796-B2 1-butyl-2-hydroxyaralkyl piperazine derivatives and the uses as anti-depression medicine thereof CSPC Zhonggi Pharmaceutical Technology (Shijiazhuang) Co. Ltd. (CN) 2012-08-28 US disclosed
US-20110183996-A1 THE 1-BUTYL-2-HYDROXYARALKYL PIPERAZINE DERIVATIVES AND THE USES AS ANTI-DEPRESSION MEDICINE THEREOF SHANGHAI INSTITUTE OF PHARMACEUTICAL INDUSTRY (CN) 2011-07-28 US disclosed
US-6864381-B2 Process for preparing acyloxybenzenesulfonates CLARIANT GMBH (DE) 2005-03-08 US disclosed
US-6822113-B2 REACTING ANHYDROUS PHENOLSULFONATES WITH CARBOXYLIC ACID DERIVATIVES BY CONTACTING THE SALT OF A PHENOLSULFONIC ACID AFTER ITS ISOLATION WITH AT LEAST ONE SUBSTANCE HAVING BASIC PROPERTIES; CONTINUOUS PROCESSING; EFFICIENCY; QUALITY CLARIANT GMBH (DE) 2004-11-23 US disclosed
US-20040198995-A1 Process for preparing acyloxybenzenesulfonates CLARIANT GMBH 2004-10-07 US disclosed
US-20040019229-A1 Process for preparing acyloxybenzenesulfonates CLARIANT GMBH 2004-01-29 US disclosed
EP-1095127-A1 NOVEL CYCLIC IMIDO BLEACH ACTIVATORS AND COMPOSITIONS CONTAINING SAME The Procter & Gamble Company (US) 2001-05-02 EP disclosed
WO-2000002990-A1 NOVEL CYCLIC IMIDO BLEACH ACTIVATORS AND COMPOSITIONS CONTAINING SAME THE PROCTER & GAMBLE COMPANY (US) 2000-01-20 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (3 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20040019229-A1 Process for preparing acyloxybenzenesulfonates AGPS, ACMSD, ARSA ALDH1A1 1959/4885POLB 340/4885KDM4E 1998/4885
US-20110183996-A1 THE 1-BUTYL-2-HYDROXYARALKYL PIPERAZINE DERIVATIVES AND THE USES AS ANTI-DEPRESSION MEDICINE THEREOF TPH2, TPH1, SLC6A4 ALDH1A1 290/4885POLB 1351/4885KDM4E 2360/4885
US-20040198995-A1 Process for preparing acyloxybenzenesulfonates TST, TYR, ACMSD ALDH1A1 943/4885POLB 190/4885KDM4E 400/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.