SCHEMBL6289352

SCHEMBL6289352

Cn1cc(Cc2ccc(F)cc2)c(=O)c2nc(C(=O)O)oc21

nearest known ligand 0.38

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
PLA2G7 Q13093 1/20 0.38
NPSR1 Q6W5P4 2/20 0.34
TP53 P04637 2/20 0.34
MAPT P10636 2/20 0.34
THRB P10828 2/20 0.34
CNR2 P34972 1/20 0.34
GPR55 Q9Y2T6 1/20 0.34
MEN1 O00255 1/20 0.34
KMT2A Q03164 1/20 0.34
MAPK14 Q16539 1/20 0.34
PPARG P37231 1/20 0.33
ADCY10 Q96PN6 1/20 0.33
EGLN1 Q9GZT9 1/20 0.32
SMN1; SMN2 Q16637 1/20 0.32
ALDH1A1 P00352 1/20 0.32
RXFP1 Q9HBX9 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6289333 0.85 LMNA (0.44) TP53MAPTTHRBCNR2MEN1
SCHEMBL6288706 0.77 CNR2 (0.40) PLA2G7TP53MAPTCNR2GPR55
SCHEMBL6289351 0.77 MMP13 (0.35) PLA2G7NPSR1TP53MAPTCNR2
SCHEMBL6288949 0.77 PHGDH (0.42) TP53MAPTALDH1A1
SCHEMBL6292166 0.75 PLA2G7 (0.38) PLA2G7TP53MAPTMEN1KMT2A
SCHEMBL6289283 0.73 MEN1 (0.43) PLA2G7TP53MAPTCNR2GPR55
SCHEMBL6289330 0.71 MMP13 (0.38) MEN1KMT2APPARGALDH1A1
SCHEMBL6292734 0.69 LMNA (0.47) TP53MAPTTHRBCNR2MEN1
SCHEMBL6476602 0.68 FPR1 (0.44) NPSR1MAPTCNR2GPR55MEN1
SCHEMBL6288785 0.68 LMNA (0.47) TP53MAPTCNR2MEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6949651-B2 Fused bicyclic metalloproteinase inhibitors WARNER-LAMBERT COMPANY (US) 2005-09-27 US disclosed
US-20040034054-A1 Fused bicyclic metalloproteinase inhibitors LINCOLN FOODSERVICE PRODUCTS INC. 2004-02-19 US disclosed
WO-2004014375-A2 FUSED BICYCLIC METALLOPROTEINASE INHIBITORS WARNER-LAMBERT COMPANY LLC (US) 2004-02-19 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20040034054-A1 Fused bicyclic metalloproteinase inhibitors MMP9, MMP1, MMP2 PLA2G7 189/4885NPSR1 2675/4885TP53 1049/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.