SCHEMBL6294222

SCHEMBL6294222

O=S(=O)(Cl)c1ccccc1-c1ccccc1Br

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CA1 P00915 2/20 0.48
CA2 P00918 2/20 0.48
CA4 P22748 2/20 0.48
CA6 P23280 2/20 0.48
PLCG1 P19174 1/20 0.45
ALDH1A1 P00352 2/20 0.41
MAPK1 P28482 1/20 0.41
HSD17B10 Q99714 1/20 0.38
TDP1 Q9NUW8 1/20 0.38
MAPT P10636 1/20 0.36
CA12 O43570 1/20 0.34
CYP2C9 P11712 1/20 0.34
CA5A P35218 1/20 0.34
CA7 P43166 1/20 0.34
CA9 Q16790 1/20 0.34
CA14 Q9ULX7 1/20 0.34
CA5B Q9Y2D0 1/20 0.34
AKR1B1 P15121 1/20 0.34
IDO1 P14902 2/20 0.33
DNMT1 P26358 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7127239 0.87 ALDH1A1 (0.48) CA1CA2CA4CA6PLCG1
SCHEMBL29540971 0.82 CA1 (0.62) CA1CA2CA4CA6PLCG1
SCHEMBL8071 0.82 CA1 (0.62) CA1CA2CA4CA6PLCG1
SCHEMBL5818974 0.81 CA2 (0.50) CA1CA2CA4CA6PLCG1
SCHEMBL7078176 0.81 CA2 (0.68) CA1CA2CA4CA6PLCG1
SCHEMBL2007711 0.76 PTPRC (0.44) CA1CA2CA4CA6ALDH1A1
SCHEMBL6291104 0.75 ALDH1A1 (0.43) ALDH1A1HSD17B10TDP1MAPTAKR1B1
SCHEMBL5679063 0.75 CA12 (0.43) CA1CA2ALDH1A1HSD17B10TDP1
SCHEMBL313390 0.74 ALDH1A1 (0.46) ALDH1A1MAPK1HSD17B10TDP1AKR1B1
SCHEMBL841244 0.74 CA2 (0.46) CA1CA2CA4CA6PLCG1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6949545-B2 Heterocyclic side chain containing, n-substituted metalloprotease inhibitors THE PROCTER & GAMBLE COMPANY (US) 2005-09-27 US disclosed
US-20040127498-A1 Heterocyclic side chain containing, n-substituted metalloprotease inhibitors THE PROCTER & GAMBLE COMPANY 2004-07-01 US disclosed
US-20030139414-A1 Heterocyclic side chain containing, n-substituted metalloprotease inhibitors THE PROCTER & GAMBLE COMPANY 2003-07-24 US disclosed
EP-1265864-A1 HETEROCYCLIC SIDE CHAIN CONTAINING, N-SUBSTITUTED METALLOPROTEASE INHIBITORS THE PROCTER & GAMBLE COMPANY (US) 2002-12-18 EP disclosed
WO-2001070691-A1 HETEROCYCLIC SIDE CHAIN CONTAINING, N-SUBSTITUTED METALLOPROTEASE INHIBITORS THE PROCTER & GAMBLE COMPANY (US) 2001-09-27 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20030139414-A1 Heterocyclic side chain containing, n-substituted metalloprotease inhibitors MME, MMP2, MMP9 CA1 485/4885CA2 325/4885CA4 472/4885
US-20040127498-A1 Heterocyclic side chain containing, n-substituted metalloprotease inhibitors MME, MMP2, MMP9 CA1 485/4885CA2 325/4885CA4 472/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.