SCHEMBL6302571

SCHEMBL6302571

CC(C)(C)OC(=O)Nc1nc2ccccc2n1C(=O)O

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TSHR P16473 3/20 0.50
ALDH1A1 P00352 1/20 0.50
BRD4 O60885 6/20 0.47
RAB9A P51151 3/20 0.47
NPC1 O15118 2/20 0.47
MEN1 O00255 2/20 0.47
KMT2A Q03164 2/20 0.47
GAA P10253 1/20 0.47
OPRM1 P35372 1/20 0.44
OPRD1 P41143 1/20 0.44
OGFRL1 Q5TC84 1/20 0.44
ACSS2 Q9NR19 1/20 0.44
KDM4E B2RXH2 4/20 0.42
CYP1A2 P05177 1/20 0.42
CYP2C9 P11712 1/20 0.42
CYP2C19 P33261 1/20 0.42
NPSR1 Q6W5P4 1/20 0.42
TDP1 Q9NUW8 1/20 0.42
POLB P06746 1/20 0.42
L3MBTL1 Q9Y468 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28680201 0.90 TSHR (0.50) TSHRALDH1A1BRD4RAB9ANPC1
SCHEMBL32671905 0.87 TSHR (0.55) TSHRALDH1A1BRD4RAB9ANPC1
SCHEMBL11177029 0.86 TSHR (0.64) TSHRALDH1A1RAB9ANPC1MEN1
SCHEMBL14920104 0.83 ACSS2 (0.41) BRD4RAB9ANPC1MEN1KMT2A
SCHEMBL11826645 0.82 TSHR (0.56) TSHRALDH1A1RAB9ANPC1MEN1
SCHEMBL11832226 0.82 ALDH1A1 (0.50) TSHRALDH1A1BRD4RAB9ANPC1
SCHEMBL11224973 0.80 RAB9A (0.51) TSHRALDH1A1RAB9ANPC1MEN1
SCHEMBL7590440 0.79 BRD4 (0.45) TSHRALDH1A1BRD4RAB9ANPC1
SCHEMBL11831949 0.78 TSHR (0.52) TSHRALDH1A1RAB9ANPC1MEN1
SCHEMBL2674793 0.76 L3MBTL1 (0.47) TSHRALDH1A1RAB9ANPC1MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3362436-B1 PROCESS FOR THE CATALYTIC DIRECTED CLEAVAGE OF AMIDE-CONTAINING COMPOUNDS UNIV ANTWERPEN (BE) 2021-06-30 EP disclosed
US-6846833-B2 Vitronectin receptor antagonist bicyclic compounds, preparation method and compositions containing same LES LABORATORIES SERVIER (FR) 2005-01-25 US disclosed
EP-1268429-B1 VITRONECTIN RECEPTOR ANTAGONIST BICYCLIC COMPOUNDS, PREPARATION METHOD AND COMPOSITIONS CONTAINING SAME SERVIER LAB (FR) 2004-08-18 EP disclosed
EP-1268429-A1 VITRONECTIN RECEPTOR ANTAGONIST BICYCLIC COMPOUNDS, PREPARATION METHOD AND COMPOSITIONS CONTAINING SAME Les Laboratoires Servier (FR) 2003-01-02 EP disclosed
WO-2001079172-A1 VITRONECTIN RECEPTOR ANTAGONIST BICYCLIC COMPOUNDS, PREPARATION METHOD AND COMPOSITIONS CONTAINING SAME LES LABORATOIRES SERVIER Departament Brevets/Fontanes (FR) 2001-10-25 WO disclosed