SCHEMBL6344199

SCHEMBL6344199

O=C1C=CC(=O)N1c1cn(-c2ccsc2)c2ccccc12

nearest known ligand 0.40

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
TLR9 Q9NR96 1/20 0.40
MGLL Q99685 11/20 0.35
MEN1 O00255 1/20 0.34
NPC1 O15118 1/20 0.34
RAB9A P51151 1/20 0.34
KMT2A Q03164 1/20 0.34
HCAR1 Q9BXC0 1/20 0.33
FAAH O00519 2/20 0.33
CHRM1 P11229 1/20 0.32
KDM4E B2RXH2 1/20 0.32
ALDH1A1 P00352 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6344247 0.83 MGLL (0.44) TLR9MGLLMEN1NPC1RAB9A
SCHEMBL6345530 0.82 MGLL (0.50) TLR9MGLLFAAHKDM4EALDH1A1
SCHEMBL4845035 0.75 PRKCB (0.45) TLR9MGLLALDH1A1
SCHEMBL6348067 0.75 TLR9 (0.40) TLR9MGLLFAAHCHRM1KDM4E
SCHEMBL4849912 0.75 HSP90AA1 (0.58) TLR9MGLLNPC1RAB9AFAAH
SCHEMBL6355781 0.71 HSP90AA1 (0.46) TLR9MGLLCHRM1
SCHEMBL28090496 0.71 MGLL (0.54) MGLLFAAHALDH1A1
SCHEMBL6345973 0.69 MGLL (0.45) TLR9MGLLMEN1KMT2AKDM4E
SCHEMBL5688433 0.69 TLR9 (0.50) TLR9MGLLKMT2AFAAHALDH1A1
SCHEMBL4847504 0.69 PRKCG (0.41) TLR9MGLL

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6849643-B2 Indazolyl-substituted pyrroline compounds as kinase inhibitors ORTHO-MCNEIL PHARMACEUTICAL, INC. (US) 2005-02-01 US disclosed