SCHEMBL6344247

SCHEMBL6344247

O=C1C=CC(=O)N1c1cn(-c2cccc(-c3ccsc3)c2)c2ccccc12

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MGLL Q99685 5/20 0.44
FAAH O00519 3/20 0.44
ALDH1A1 P00352 1/20 0.44
HSP90AA1 P07900 1/20 0.44
PKM P14618 1/20 0.44
HTT P42858 1/20 0.44
ATM Q13315 1/20 0.44
ALOX5 P09917 1/20 0.41
PTPRC P08575 1/20 0.35
GLO1 Q04760 1/20 0.35
CYP2E1 P05181 1/20 0.35
CYP2A6 P11509 1/20 0.35
CYP2B6 P20813 1/20 0.35
WNK1 Q9H4A3 1/20 0.34
COMT P21964 2/20 0.33
PRKDC P78527 1/20 0.33
TLR9 Q9NR96 1/20 0.33
PRMT6 Q96LA8 1/20 0.32
KDR P35968 1/20 0.32
MEN1 O00255 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6344199 0.83 TLR9 (0.40) MGLLFAAHALDH1A1TLR9MEN1
SCHEMBL6345530 0.77 MGLL (0.50) MGLLFAAHALDH1A1HSP90AA1PKM
SCHEMBL3785977 0.73 ALOX5 (0.40) ALOX5PTPRCGLO1WNK1PRKDC
SCHEMBL4849912 0.73 HSP90AA1 (0.58) MGLLFAAHALDH1A1HSP90AA1TLR9
SCHEMBL4845035 0.70 PRKCB (0.45) MGLLALDH1A1HTTCYP2E1CYP2A6
SCHEMBL6355781 0.69 HSP90AA1 (0.46) MGLLHSP90AA1PKMTLR9
SCHEMBL6348067 0.68 TLR9 (0.40) MGLLFAAHALDH1A1TLR9
SCHEMBL6345973 0.68 MGLL (0.45) MGLLALDH1A1HSP90AA1HTTCYP2A6
SCHEMBL17502096 0.66 MPI (0.60) ALDH1A1HSP90AA1PKMNPC1RAB9A
SCHEMBL3179484 0.64 MGLL (0.88) MGLLFAAHALDH1A1HSP90AA1PKM

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6849643-B2 Indazolyl-substituted pyrroline compounds as kinase inhibitors ORTHO-MCNEIL PHARMACEUTICAL, INC. (US) 2005-02-01 US disclosed