SCHEMBL635229

SCHEMBL635229

CCN(CC)c1ccc(P(c2ccc(N(CC)CC)cc2)c2ccc3ccccc3c2-c2c(P(c3ccc(N(CC)CC)cc3)c3ccc(N(CC)CC)cc3)ccc3ccccc23)cc1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 5/20 0.42
KMT2A Q03164 5/20 0.42
NPC1 O15118 2/20 0.42
ACHE P22303 4/20 0.41
KDM1A O60341 1/20 0.40
PLK1 P53350 1/20 0.39
CNR2 P34972 2/20 0.37
BCHE P06276 2/20 0.36
ALDH1A1 P00352 3/20 0.36
MAPK1 P28482 3/20 0.36
TDP1 Q9NUW8 2/20 0.36
L3MBTL1 Q9Y468 2/20 0.36
TSHR P16473 2/20 0.36
PSMD14 O00487 1/20 0.36
CYP3A4 P08684 1/20 0.36
RECQL P46063 1/20 0.36
GFER P55789 1/20 0.36
NPY5R Q15761 1/20 0.36
TERT O14746 1/20 0.36
RAB9A P51151 2/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30894434 1.00 MEN1 (0.42) MEN1KMT2ANPC1ACHEKDM1A
SCHEMBL636417 0.86 NPC1 (0.41) MEN1KMT2ANPC1ACHEKDM1A
SCHEMBL11911370 0.85 TDP1 (0.40) MEN1KMT2ANPC1ACHEKDM1A
SCHEMBL635353 0.83 ALOX5 (0.40) MEN1KMT2ANPC1KDM1ACNR2
SCHEMBL15094120 0.82 CYP1A2 (0.38) KMT2AALDH1A1TDP1TSHRCYP3A4
Hydrochloric Acid SCHEMBL16561297 0.81 MAPT (0.40) MEN1KMT2ANPC1KDM1ACNR2
SCHEMBL29361524 0.78 MAPT (0.39) MEN1KMT2ANPC1ALDH1A1MAPK1
SCHEMBL29176 0.78 MAPT (0.39) MEN1KMT2ANPC1ALDH1A1MAPK1
SCHEMBL146878 0.77 ALDH1A1 (0.44) ALDH1A1MAPK1TDP1TSHRCYP3A4
SCHEMBL5107 0.77 ALDH1A1 (0.44) ALDH1A1MAPK1TDP1TSHRCYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 36 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1927596-B9 DIPHOSPHINE LIGAND AND TRANSITION METAL COMPLEX USING THE SAME TAKEDA PHARMACEUTICAL (JP) 2013-05-15 EP claimed
EP-1927596-B1 DIPHOSPHINE LIGAND AND TRANSITION METAL COMPLEX USING THE SAME TAKEDA PHARMACEUTICAL (JP) 2012-08-01 EP claimed
EP-2420507-A1 Diphosphine ligand and transition metal complex using the same Takeda Pharmaceutical Company Limited (JP) 2012-02-22 EP claimed
US-20090270635-A1 Diphosphine Ligand and Transition Metal Complex Using the Same TAKEDA PHARMACEUTICAL COMPANY LIMITED 2009-10-29 US claimed
EP-1927596-A1 DIPHOSPHINE LIGAND AND TRANSITION METAL COMPLEX USING THE SAME Takeda Pharmaceutical Company Limited (JP) 2008-06-04 EP claimed
US-12129249-B2 Method for producing optically active compound DAY ONE BIOPHARMACEUTICALS, INC. (US) 2024-10-29 US disclosed
EP-4406609-A2 METHOD FOR PRODUCING OPTICALLY ACTIVE COMPOUND Day One Biopharmaceuticals, Inc. (US) 2024-07-31 EP disclosed
CN-118005619-A Process for producing heterocyclic compound 武田药品工业株式会社 2024-05-10 CN disclosed
US-20210347769-A1 METHOD FOR PRODUCING OPTICALLY ACTIVE COMPOUND DAY ONE BIOPHARMACEUTICALS, INC. 2021-11-11 US disclosed
US-10988469-B2 Method for producing optically active compound DOT THERAPEUTICS-1, INC. (US) 2021-04-27 US disclosed
US-20200317659-A1 METHOD FOR PRODUCING OPTICALLY ACTIVE COMPOUND DAY ONE BIOPHARMACEUTICALS, INC. 2020-10-08 US disclosed
US-10710989-B2 Method for producing heterocyclic compound TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2020-07-14 US disclosed
EP-1927596-B9 DIPHOSPHINE LIGAND AND TRANSITION METAL COMPLEX USING THE SAME TAKEDA PHARMACEUTICAL (JP) 2013-05-15 EP disclosed
EP-1927596-B1 DIPHOSPHINE LIGAND AND TRANSITION METAL COMPLEX USING THE SAME TAKEDA PHARMACEUTICAL (JP) 2012-08-01 EP disclosed
EP-2420507-A1 Diphosphine ligand and transition metal complex using the same Takeda Pharmaceutical Company Limited (JP) 2012-02-22 EP disclosed
EP-2420507-A1 Diphosphine ligand and transition metal complex using the same Takeda Pharmaceutical Company Limited (JP) 2012-02-22 EP disclosed
US-20090270635-A1 Diphosphine Ligand and Transition Metal Complex Using the Same TAKEDA PHARMACEUTICAL COMPANY LIMITED 2009-10-29 US disclosed
US-20090270635-A1 Diphosphine Ligand and Transition Metal Complex Using the Same TAKEDA PHARMACEUTICAL COMPANY LIMITED 2009-10-29 US disclosed
EP-1927596-A1 DIPHOSPHINE LIGAND AND TRANSITION METAL COMPLEX USING THE SAME Takeda Pharmaceutical Company Limited (JP) 2008-06-04 EP disclosed
EP-1927596-A1 DIPHOSPHINE LIGAND AND TRANSITION METAL COMPLEX USING THE SAME Takeda Pharmaceutical Company Limited (JP) 2008-06-04 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (6 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-10988469-B2 Method for producing optically active compound DHPS, QDPR, SPR MEN1 1696/4885KMT2A 504/4885NPC1 2691/4885
US-20200317659-A1 METHOD FOR PRODUCING OPTICALLY ACTIVE COMPOUND DHPS, QDPR, SPR MEN1 1696/4885KMT2A 504/4885NPC1 2691/4885
US-12129249-B2 Method for producing optically active compound DHPS, QDPR, SPR MEN1 1696/4885KMT2A 504/4885NPC1 2691/4885
US-10710989-B2 Method for producing heterocyclic compound APP, THOP1, TALDO1 MEN1 1683/4885KMT2A 2686/4885NPC1 635/4885
US-20090270635-A1 Diphosphine Ligand and Transition Metal Complex Using the Same MVD, C5, C1S MEN1 658/4885KMT2A 1029/4885NPC1 4580/4885
US-20210347769-A1 METHOD FOR PRODUCING OPTICALLY ACTIVE COMPOUND DHPS, QDPR, SPR MEN1 1696/4885KMT2A 504/4885NPC1 2691/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.