SCHEMBL6366012

SCHEMBL6366012

O=c1cc[nH]c2ccccc12.[NaH]

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.53
CCR8 P51685 1/20 0.48
HSD17B10 Q99714 3/20 0.47
KMT2A Q03164 1/20 0.46
AHR P35869 2/20 0.44
TRPA1 O75762 1/20 0.44
CA1 P00915 1/20 0.44
CA2 P00918 1/20 0.44
ITGB2 P05107 1/20 0.44
ICAM1 P05362 1/20 0.44
ITGAL P20701 1/20 0.44
CA4 P22748 1/20 0.44
CA6 P23280 1/20 0.44
ADK P55263 1/20 0.44
KDM4E B2RXH2 4/20 0.44
CYP1A2 P05177 2/20 0.44
GAA P10253 2/20 0.44
PARP1 P09874 1/20 0.43
CYP3A4 P08684 1/20 0.43
CYP2D6 P10635 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10031 0.98 ALDH1A1 (0.55) ALDH1A1CCR8HSD17B10KMT2AAHR
Hydrochloric Acid SCHEMBL3646722 0.95 ALDH1A1 (0.53) ALDH1A1CCR8HSD17B10KMT2AAHR
Benzene SCHEMBL28794130 0.95 ALDH1A1 (0.53) ALDH1A1CCR8HSD17B10KMT2AAHR
Hydrochloric Acid SCHEMBL3397919 0.95 ALDH1A1 (0.53) ALDH1A1CCR8HSD17B10KMT2AAHR
SCHEMBL20677769 0.95 ALDH1A1 (0.53) ALDH1A1CCR8HSD17B10KMT2AAHR
Hydrochloric Acid SCHEMBL29744420 0.95 ALDH1A1 (0.53) ALDH1A1CCR8HSD17B10KMT2AAHR
Iodide SCHEMBL7508631 0.95 ALDH1A1 (0.53) ALDH1A1CCR8HSD17B10KMT2AAHR
Fluoride SCHEMBL4741374 0.95 ALDH1A1 (0.53) ALDH1A1CCR8HSD17B10KMT2AAHR
SCHEMBL18900583 0.84 FKBP5 (0.44) ALDH1A1HSD17B10KMT2AAHRKDM4E
Fumaric Acid SCHEMBL4611816 0.83 HTR1A (0.47) ALDH1A1HSD17B10KMT2AAHRKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20050075334-A1 8-(1H-Benzimidazol-2-ylsulfanyl)-4(1H)-quinolinone derivatives; jun N-terminal kinase inhibitors; Alzheimer*s, Parkinson*s, and Huntington*s disease; amyotrophic lateral sclerosis, antiepileptic agents; hemorrhage, seizures, traumatic brain injuries or haemorrhaging strokes ASTRAZENECA AB (SE) 2005-04-07 US disclosed
EP-1458712-A2 NOVEL COMPOUNDS AstraZeneca AB (SE) 2004-09-22 EP disclosed
WO-2003051277-A2 NOVEL COMPOUNDS ASTRAZENECA AB (SE) 2003-06-26 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20050075334-A1 8-(1H-Benzimidazol-2-ylsulfanyl)-4(1H)-quinolinone derivatives; jun N-terminal kinase inhibitors; Alzheimer*s, Parkinson*s, and Huntington*s disease; amyotrophic lateral sclerosis, antiepileptic agents; hemorrhage, seizures, traumatic brain injuries or haemorrhaging strokes PARK7, HYPK, BCL2A1 ALDH1A1 2650/4885CCR8 2234/4885HSD17B10 3012/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.