SCHEMBL6396359

SCHEMBL6396359

C=C(C(=O)OC)C(OC(C)=O)c1ccccc1

nearest known ligand 0.57

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.57
CYP3A4 P08684 1/20 0.57
TSHR P16473 1/20 0.49
HSD17B10 Q99714 2/20 0.45
HPGD P15428 1/20 0.45
KMT2A Q03164 1/20 0.43
GLS O94925 3/20 0.43
MAPK1 P28482 1/20 0.43
CASP3 P42574 1/20 0.41
CASP2 P42575 1/20 0.41
CASP7 P55210 1/20 0.41
CASP6 P55212 1/20 0.41
CASP8 Q14790 1/20 0.41
KDM4E B2RXH2 1/20 0.41
MAPT P10636 1/20 0.41
CASP1 P29466 1/20 0.41
HTT P42858 1/20 0.41
GAA P10253 2/20 0.40
SMN1; SMN2 Q16637 1/20 0.40
L3MBTL1 Q9Y468 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27528908 0.89 KMT2A (0.44) ALDH1A1CYP3A4TSHRHPGDKMT2A
SCHEMBL17221835 0.86 ALDH1A1 (0.41) ALDH1A1CYP3A4TSHRHSD17B10MAPK1
SCHEMBL4014931 0.85 ALDH1A1 (0.62) ALDH1A1CYP3A4TSHRHSD17B10HPGD
SCHEMBL12571904 0.84 CYP1A2 (0.44) ALDH1A1CYP3A4TSHRHPGDMAPK1
SCHEMBL24091673 0.84 RAB9A (0.44) ALDH1A1CYP3A4TSHRHPGDKMT2A
SCHEMBL29473539 0.83 ALDH1A1 (0.53) ALDH1A1CYP3A4TSHRHSD17B10HPGD
SCHEMBL4013821 0.83 ALDH1A1 (0.53) ALDH1A1CYP3A4TSHRHSD17B10HPGD
SCHEMBL19031592 0.83 KDM4E (0.44) ALDH1A1CYP3A4TSHRKDM4EGAA
SCHEMBL19031584 0.83 ALDH1A1 (0.39) ALDH1A1CYP3A4HPGDKMT2ASMN1; SMN2
SCHEMBL19031506 0.83 CYP2D6 (0.42) ALDH1A1CYP3A4TSHRHSD17B10KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 21 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20050006246-A1 Nitrogen atom transfer YUDIN ANDREI K (CA) 2005-01-13 US claimed
WO-2003010361-A2 NITROGEN ATOM TRANSFER YLEKTRA INC. (CA) 2003-02-06 WO claimed
EP-3440051-B1 NEUROPEPTIDE S RECEPTOR (NPSR) AGONISTS RES TRIANGLE INST (US) 2024-03-20 EP disclosed
US-20210380635-A1 COMPOSITIONS AND METHODS FOR PROTEIN LABELING, MODIFICATION, ANALYSIS, AND TARGETED DELIVERY NATIONAL INSTITUTES OF HEALTH (NIH), U.S. DEPT. OF HEALTH AND HUMAN SERVICES (DHHS), U.S. GOVERNMENT 2021-12-09 US disclosed
US-11186678-B2 Radical cascade-enabled synthesis of precision polymers with complex main-chain structures TRUSTEES OF BOSTON COLLEGE (US) 2021-11-30 US disclosed
US-11142546-B2 Neuropeptide S receptor (NPSR) agonists RESEARCH TRIANGLE INSTITUTE (US) 2021-10-12 US disclosed
US-20200216610-A1 RADICAL CASCADE-ENABLED SYNTHESIS OF PRECISION POLYMERS WITH COMPLEX MAIN-CHAIN STRUCTURES TRUSTEES OF BOSTON COLLEGE (US) 2020-07-09 US disclosed
WO-2019060809-A1 INHIBITORS OF PSEUDOMONAS AERUGINOSA VIRULENCE CHANNEL THERAPEUTICS, INC. (US) 2019-03-28 WO disclosed
US-20190092809-A1 NEUROPEPTIDE S RECEPTOR (NPSR) AGONISTS NATIONAL INSTITUTES OF HEALTH (NIH), U.S. DEPT. OF HEALTH AND HUMAN SERVICES (DHHS), U.S. GOVERNMENT 2019-03-28 US disclosed
EP-3440051-A1 NEUROPEPTIDE S RECEPTOR (NPSR) AGONISTS Research Triangle Institute (US) 2019-02-13 EP disclosed
WO-2017176461-A1 NEUROPEPTIDE S RECEPTOR (NPSR) AGONISTS RESEARCH TRIANGLE INSTITUTE (US) 2017-10-12 WO disclosed
WO-2017109795-A1 NOVEL COMPOUNDS USEFUL AS POTENTIAL INSECT ANTIFEEDANT AND A PROCESS FOR THE PREPARATION THEREOF COUNCIL OF SCIENTIFIC & INDUSTRIAL RESEARCH (IN) 2017-06-29 WO disclosed
US-9249139-B2 Indolizinone based derivatives as potential phosphodiesterase 3 (PDE3) inhibitors and a process for the preparation thereof COUNCIL OF SCIENTIFIC & INDUSTRIAL RESEARCH (IN) 2016-02-02 US disclosed
US-20150045556-A1 PROCESSES FOR THE PREPARATION OF PERIPHERAL OPIOID ANTAGONIST COMPOUNDS AND INTERMEDIATES THERETO DOLLE ROLAND E (US) 2015-02-12 US disclosed
WO-2013012871-A1 PROCESSES FOR THE PREPARATION OF PERIPHERAL OPIOID ANTAGONIST COMPOUNDS AND INTERMEDIATES THERETO ADOLOR CORPORATION (US) 2013-01-24 WO disclosed
US-20070203224-A1 SMALL-MOLECULES FOR TREATING CANCER AND ABNORMAL CELL PROLIFERATION DISORDERS UNIVERSITY OF SOUTHERN CALIFORNIA 2007-08-30 US disclosed
US-20070203224-A1 SMALL-MOLECULES FOR TREATING CANCER AND ABNORMAL CELL PROLIFERATION DISORDERS UNIVERSITY OF SOUTHERN CALIFORNIA 2007-08-30 US disclosed
WO-2007081966-A2 SMALL MOLECULES FOR TREATING CANCER AND ABNORMAL CELL PROLIFERATION DISORDERS UNIVERSITY OF SOUTHERN CALIFORNIA (US) 2007-07-19 WO disclosed
US-20050006246-A1 Nitrogen atom transfer YUDIN ANDREI K (CA) 2005-01-13 US disclosed
WO-2003010361-A2 NITROGEN ATOM TRANSFER YLEKTRA INC. (CA) 2003-02-06 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (4 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20150045556-A1 PROCESSES FOR THE PREPARATION OF PERIPHERAL OPIOID ANTAGONIST COMPOUNDS AND INTERMEDIATES THERETO OPRK1, OPRM1, OPRD1 ALDH1A1 2714/4885CYP3A4 137/4885TSHR 985/4885
US-20190092809-A1 NEUROPEPTIDE S RECEPTOR (NPSR) AGONISTS NPSR1, GRPR, NPBWR1 ALDH1A1 4747/4885CYP3A4 3917/4885TSHR 62/4885
US-20210380635-A1 COMPOSITIONS AND METHODS FOR PROTEIN LABELING, MODIFICATION, ANALYSIS, AND TARGETED DELIVERY PTMS, SRMS, CHAMP1 ALDH1A1 3049/4885CYP3A4 3746/4885TSHR 3028/4885
US-11142546-B2 Neuropeptide S receptor (NPSR) agonists NPSR1, GRPR, NPBWR1 ALDH1A1 4747/4885CYP3A4 3917/4885TSHR 62/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.