Leucine

Leucine

SCHEMBL6415294

CC(C)C[C@H](N)C(=O)O.O=C(O)CCN[C@H](CCc1ccccc1)C(=O)O

nearest known ligand 0.48

Full drug profile on Sugi Atlas →

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
LTA4H P09960 1/20 0.46
GRIK1 P39086 1/20 0.46
MMP3 P08254 1/20 0.46
GGT1 P19440 1/20 0.45
ERAP2 Q6P179 3/20 0.45
ERAP1 Q9NZ08 3/20 0.45
LNPEP Q9UIQ6 1/20 0.45
ANPEP P15144 2/20 0.44
RNPEP Q9H4A4 1/20 0.43
DNPEP Q9ULA0 1/20 0.43
SLC7A5 Q01650 1/20 0.43
SLC1A1 P43005 1/20 0.42
MME P08473 1/20 0.41
LMNA P02545 1/20 0.41
PKM P14618 1/20 0.41
IL1RN P18510 2/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Leucine SCHEMBL7383434 0.91 SLC7A5 (0.41) LTA4HGRIK1MMP3GGT1ERAP2
Leucine SCHEMBL7375203 0.91 MMP3 (0.46) LTA4HMMP3ERAP2ERAP1LNPEP
Leucine SCHEMBL7383856 0.91 MMP8 (0.44) LTA4HGRIK1MMP3ERAP2ERAP1
Leucine SCHEMBL7382855 0.90 LMNA (0.45) LTA4HMMP3ERAP2ERAP1LNPEP
Leucine SCHEMBL7378736 0.89 MASP2 (0.43) LTA4HMMP3ERAP2ERAP1LNPEP
Homophenylalanine SCHEMBL7383933 0.89 GGT1 (0.50) LTA4HGRIK1GGT1SLC7A5MME
Alanine SCHEMBL7382718 0.89 GGT1 (0.50) MMP3GGT1MMELMNAPKM
Glutamic Acid SCHEMBL7375280 0.88 GGT1 (0.49) LTA4HGRIK1GGT1SLC7A5SLC1A1
Asparagine SCHEMBL7375839 0.87 GGT1 (0.46) GRIK1GGT1SLC7A5SLC1A1MME
Serine SCHEMBL7384366 0.86 GGT1 (0.48) LTA4HGRIK1GGT1SLC7A5MME

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 9 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20050020607-A1 Statin-MMP inhibitor combinations NEWTON ROGER SCHOFIELD (US) 2005-01-27 US disclosed
EP-1098662-A2 COADMINISTRATION OF ACAT AND MMP INHIBITORS FOR THE TREATMENT OF ATHEROSCLEROTIC LESIONS WARNER-LAMBERT COMPANY (US) 2001-05-16 EP disclosed
EP-1063991-A1 STATIN-MATRIX METALLOPROTEINASE INHIBITOR COMBINATIONS WARNER-LAMBERT COMPANY LLC (US) 2001-01-03 EP disclosed
EP-1047450-A1 ACE INHIBITOR-MMP INHIBITOR COMBINATIONS WARNER-LAMBERT COMPANY (US) 2000-11-02 EP disclosed
WO-2000004892-A2 COADMINISTRATION OF ACAT AND MMP INHIBITORS FOR THE TREATMENT OF ATHEROSCLEROTIC LESIONS WARNER-LAMBERT COMPANY (US) 2000-02-03 WO disclosed
EP-0946166-A1 USE OF MATRIX METALLOPROTEINASE INHIBITORS FOR TREATING NEUROLOGICAL DISORDERS AND PROMOTING WOUND HEALING WARNER-LAMBERT COMPANY (US) 1999-10-06 EP disclosed
WO-1999047138-A1 STATIN-MATRIX METALLOPROTEINASE INHIBITOR COMBINATIONS WARNER-LAMBERT COMPANY (US) 1999-09-23 WO disclosed
WO-1999032150-A1 ACE INHIBITOR-MMP INHIBITOR COMBINATIONS WARNER-LAMBERT COMPANY (US) 1999-07-01 WO disclosed
WO-1998026773-A1 USE OF MATRIX METALLOPROTEINASE INHIBITORS FOR TREATING NEUROLOGICAL DISORDERS AND PROMOTING WOUND HEALING WARNER-LAMBERT COMPANY (US) 1998-06-25 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20050020607-A1 Statin-MMP inhibitor combinations MMP9, TIMP3, MMP3 LTA4H 378/4885GRIK1 3971/4885MMP3 3/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.