SCHEMBL6416161

SCHEMBL6416161

COc1ccc(O)c(NC(=O)C(=O)Nc2cc(Cl)cc(Cl)c2O)c1

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 6/20 0.52
KMT2A Q03164 6/20 0.52
L3MBTL1 Q9Y468 1/20 0.52
NPC1 O15118 2/20 0.46
RAB9A P51151 1/20 0.46
KCNMA1 Q12791 4/20 0.46
KDM4E B2RXH2 2/20 0.44
HIF1A Q16665 1/20 0.44
TDP1 Q9NUW8 1/20 0.44
HSPA5 P11021 1/20 0.44
FADS1 O60427 1/20 0.43
MAPT P10636 3/20 0.43
LMNA P02545 2/20 0.43
THRB P10828 1/20 0.43
MCL1 Q07820 1/20 0.42
POLB P06746 2/20 0.42
KCNH2 Q12809 1/20 0.42
GAA P10253 1/20 0.42
ALDH1A1 P00352 1/20 0.41
ACLY P53396 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6408135 0.84 KCNMA1 (0.55) MEN1KMT2AKCNMA1HSPA5POLB
SCHEMBL6410312 0.80 KCNMA1 (0.52) KCNMA1KDM4EHIF1ATDP1HSPA5
SCHEMBL6415342 0.80 HSPA5 (0.47) MEN1KMT2AKCNMA1HSPA5MAPT
SCHEMBL6410292 0.80 HSPA5 (0.62) MEN1KMT2AKDM4EHIF1AHSPA5
SCHEMBL6414640 0.78 ACLY (0.49) MEN1KMT2AL3MBTL1KCNMA1KDM4E
SCHEMBL6407663 0.77 NPC1 (0.50) MEN1KMT2ANPC1RAB9AKCNMA1
SCHEMBL6411984 0.77 HSPA5 (0.47) MEN1KMT2ANPC1RAB9AKCNMA1
SCHEMBL6409044 0.77 KMT2A (0.50) MEN1KMT2ARAB9AKCNMA1KDM4E
SCHEMBL6415355 0.76 HSPA5 (0.44) MEN1KMT2AKCNMA1HSPA5MAPT
SCHEMBL6408459 0.76 ACLY (0.59) KCNMA1KDM4EACLY

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20050124667-A1 Oxamide inhibitors of plasminogen activator inhibitor-1 CEREP SA (FR) 2005-06-09 US claimed
US-20050124667-A1 Oxamide inhibitors of plasminogen activator inhibitor-1 CEREP SA (FR) 2005-06-09 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20050124667-A1 Oxamide inhibitors of plasminogen activator inhibitor-1 SERPINE1, SERPINC1, SERPINB1 MEN1 1009/4885KMT2A 3936/4885L3MBTL1 1784/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.