SCHEMBL6415342

SCHEMBL6415342

Nc1ccc(O)c(NC(=O)C(=O)Nc2cc(Cl)cc(Cl)c2O)c1

nearest known ligand 0.47

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
HSPA5 P11021 1/20 0.47
KCNMA1 Q12791 11/20 0.43
POLB P06746 1/20 0.43
CA1 P00915 1/20 0.42
CA2 P00918 1/20 0.42
CHRNA7 P36544 1/20 0.39
MEN1 O00255 1/20 0.38
MAPT P10636 1/20 0.38
KMT2A Q03164 1/20 0.38
STAT3 P40763 1/20 0.38
HSD17B10 Q99714 2/20 0.38
SMN1; SMN2 Q16637 1/20 0.38
NPSR1 Q6W5P4 1/20 0.38
MAPK1 P28482 1/20 0.37
HDAC1 Q13547 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6408135 0.88 KCNMA1 (0.55) HSPA5KCNMA1POLBCHRNA7MEN1
SCHEMBL6410312 0.83 KCNMA1 (0.52) HSPA5KCNMA1POLBCHRNA7STAT3
SCHEMBL6410292 0.83 HSPA5 (0.62) HSPA5POLBCA1CA2MEN1
SCHEMBL6412941 0.82 CA1 (0.57) CA1CA2MAPT
SCHEMBL6414640 0.82 ACLY (0.49) HSPA5KCNMA1POLBCA1CA2
SCHEMBL6407663 0.81 NPC1 (0.50) HSPA5KCNMA1POLBMEN1MAPT
SCHEMBL6415355 0.80 HSPA5 (0.44) HSPA5KCNMA1POLBMEN1MAPT
SCHEMBL6408459 0.80 ACLY (0.59) KCNMA1HDAC1
SCHEMBL6416161 0.80 MEN1 (0.52) HSPA5KCNMA1POLBMEN1MAPT
SCHEMBL6417211 0.80 CHRNA7 (0.63) HSPA5KCNMA1CHRNA7MEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20050124667-A1 Oxamide inhibitors of plasminogen activator inhibitor-1 CEREP SA (FR) 2005-06-09 US claimed
US-20050124667-A1 Oxamide inhibitors of plasminogen activator inhibitor-1 CEREP SA (FR) 2005-06-09 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20050124667-A1 Oxamide inhibitors of plasminogen activator inhibitor-1 SERPINE1, SERPINC1, SERPINB1 HSPA5 4261/4885KCNMA1 2149/4885POLB 2207/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.