SCHEMBL6415355

SCHEMBL6415355

N#Cc1ccc(O)c(NC(=O)C(=O)Nc2cc(Cl)cc(Cl)c2O)c1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HSPA5 P11021 1/20 0.44
GPR35 Q9HC97 2/20 0.43
TMPRSS4 Q9NRS4 2/20 0.43
P2RX1 P51575 1/20 0.41
KCNMA1 Q12791 4/20 0.40
POLB P06746 1/20 0.40
MEN1 O00255 2/20 0.40
KMT2A Q03164 2/20 0.40
CXCR2 P25025 2/20 0.40
CXCR1 P25024 1/20 0.39
LMNA P02545 1/20 0.38
MAPT P10636 1/20 0.38
TSHR P16473 1/20 0.38
HTT P42858 1/20 0.38
NLRP3 Q96P20 1/20 0.38
PDK1 Q15118 1/20 0.38
PDK2 Q15119 1/20 0.38
PDK3 Q15120 1/20 0.38
PDK4 Q16654 1/20 0.38
CYP1A2 P05177 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6408135 0.84 KCNMA1 (0.55) HSPA5KCNMA1POLBMEN1KMT2A
SCHEMBL6410312 0.80 KCNMA1 (0.52) HSPA5P2RX1KCNMA1POLBACLY
SCHEMBL6415342 0.80 HSPA5 (0.47) HSPA5KCNMA1POLBMEN1KMT2A
SCHEMBL6410292 0.80 HSPA5 (0.62) HSPA5POLBMEN1KMT2ALMNA
SCHEMBL6414640 0.78 ACLY (0.49) HSPA5GPR35KCNMA1POLBMEN1
SCHEMBL6407663 0.77 NPC1 (0.50) HSPA5KCNMA1POLBMEN1KMT2A
SCHEMBL4358673 0.77 LMNA (0.64) HSPA5TMPRSS4POLBMEN1KMT2A
SCHEMBL6416161 0.76 MEN1 (0.52) HSPA5KCNMA1POLBMEN1KMT2A
SCHEMBL6412941 0.76 CA1 (0.57) MAPT
SCHEMBL6408459 0.76 ACLY (0.59) KCNMA1ACLY

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20050124667-A1 Oxamide inhibitors of plasminogen activator inhibitor-1 CEREP SA (FR) 2005-06-09 US claimed
US-20050124667-A1 Oxamide inhibitors of plasminogen activator inhibitor-1 CEREP SA (FR) 2005-06-09 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20050124667-A1 Oxamide inhibitors of plasminogen activator inhibitor-1 SERPINE1, SERPINC1, SERPINB1 HSPA5 4261/4885GPR35 3140/4885TMPRSS4 191/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.