SCHEMBL64196

SCHEMBL64196

CC(C)(C)[Si](C)(C)OCC1C(C(=O)O)=C(c2ccc(OCCOc3c(Cl)cccc3Cl)cc2)CCN1C(=O)OCc1ccccc1

nearest known ligand 0.36

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
GHSR Q92847 3/20 0.36
CHRM5 P08912 1/20 0.36
CHRM1 P11229 1/20 0.36
PTGDR2 Q9Y5Y4 4/20 0.35
KDM4E B2RXH2 1/20 0.34
LMNA P02545 1/20 0.34
ABCB1 P08183 1/20 0.34
PPARA Q07869 1/20 0.34
PARP1 P09874 1/20 0.33
AOC3 Q16853 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL78781 0.93 KDM4E (0.36) GHSRCHRM5CHRM1PTGDR2KDM4E
SCHEMBL64456 0.93 PPARG (0.39) GHSRCHRM5CHRM1PTGDR2KDM4E
SCHEMBL10289284 0.88 PPARA (0.36) GHSRCHRM5CHRM1PTGDR2KDM4E
SCHEMBL78412 0.86 PPARG (0.39) CHRM5CHRM1PTGDR2KDM4ELMNA
SCHEMBL64503 0.85 PPARA (0.33) GHSRCHRM5CHRM1PTGDR2KDM4E
SCHEMBL78724 0.83 KDM4E (0.34) CHRM5CHRM1PTGDR2KDM4ELMNA
SCHEMBL65298 0.83 CHRM5 (0.35) CHRM5CHRM1
SCHEMBL64061 0.82 CHRM2 (0.38) GHSRCHRM5CHRM1PARP1
SCHEMBL64233 0.81 CHRM5 (0.35) CHRM5CHRM1PTGDR2KDM4ELMNA
SCHEMBL80037 0.81 ITGB3 (0.32) PTGDR2KDM4ELMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8129538-B1 Renin inhibitors TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2012-03-06 US disclosed
US-8129538-B1 Renin inhibitors TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2012-03-06 US disclosed