SCHEMBL78781

SCHEMBL78781

CCOC(=O)C1=C(c2ccc(OCCOc3c(Cl)cccc3Cl)cc2)CCN(C(=O)OCc2ccccc2)C1CO[Si](C)(C)C(C)(C)C

nearest known ligand 0.36

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 1/20 0.36
LMNA P02545 1/20 0.36
TP53 P04637 1/20 0.34
POLB P06746 1/20 0.34
SMN1; SMN2 Q16637 1/20 0.34
CHRM5 P08912 2/20 0.34
CHRM1 P11229 2/20 0.34
ESR1 P03372 1/20 0.34
ESR2 Q92731 1/20 0.34
GHSR Q92847 1/20 0.33
PTGDR2 Q9Y5Y4 4/20 0.33
L3MBTL1 Q9Y468 1/20 0.33
LTA4H P09960 1/20 0.33
ABCB1 P08183 1/20 0.33
CHRM2 P08172 1/20 0.33
CHRM4 P08173 1/20 0.33
CHRM3 P20309 1/20 0.33
DGAT1 O75907 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL78412 0.93 PPARG (0.39) KDM4ELMNATP53POLBSMN1; SMN2
SCHEMBL64196 0.93 GHSR (0.36) KDM4ELMNACHRM5CHRM1GHSR
SCHEMBL65298 0.91 CHRM5 (0.35) TP53POLBCHRM5CHRM1ESR1
SCHEMBL66854 0.86 CHRM2 (0.38) KDM4ELMNATP53POLBSMN1; SMN2
SCHEMBL64456 0.86 PPARG (0.39) KDM4ELMNASMN1; SMN2CHRM5CHRM1
SCHEMBL64233 0.84 CHRM5 (0.35) KDM4ELMNATP53POLBSMN1; SMN2
SCHEMBL65813 0.84 PPARG (0.40) KDM4ETP53CHRM5CHRM1L3MBTL1
SCHEMBL78622 0.83 SMN1; SMN2 (0.38) POLBSMN1; SMN2CHRM5CHRM1CHRM2
SCHEMBL91270 0.81 PPARG (0.38) KDM4ELMNATP53POLBSMN1; SMN2
SCHEMBL78724 0.81 KDM4E (0.34) KDM4ELMNACHRM5CHRM1PTGDR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8129538-B1 Renin inhibitors TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2012-03-06 US disclosed