SCHEMBL65298

SCHEMBL65298

CCOC(=O)C1=C(c2ccc(OCCOc3c(Cl)cccc3Cl)cc2)CCN(C(=O)O)C1CO[Si](C)(C)C(C)(C)C

nearest known ligand 0.35

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
CHRM5 P08912 2/20 0.35
CHRM1 P11229 2/20 0.35
CYP3A4 P08684 1/20 0.34
KCNH2 Q12809 1/20 0.33
HRH3 Q9Y5N1 1/20 0.33
GRIN2C Q14957 1/20 0.32
ESR1 P03372 1/20 0.32
ESR2 Q92731 1/20 0.32
HRH2 P25021 2/20 0.32
HRH1 P35367 2/20 0.32
POLB P06746 1/20 0.32
MAPT P10636 2/20 0.32
TP53 P04637 1/20 0.32
TDP1 Q9NUW8 1/20 0.32
L3MBTL1 Q9Y468 1/20 0.32
DHFR P00374 1/20 0.31
CHRM2 P08172 1/20 0.31
CHRM4 P08173 1/20 0.31
CHRM3 P20309 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL65813 0.92 PPARG (0.40) CHRM5CHRM1KCNH2HRH3HRH2
SCHEMBL78781 0.91 KDM4E (0.36) CHRM5CHRM1ESR1ESR2POLB
SCHEMBL64196 0.83 GHSR (0.36) CHRM5CHRM1
SCHEMBL64034 0.80 CHRM5 (0.38) CHRM5CHRM1CYP3A4POLBMAPT
SCHEMBL64233 0.76 CHRM5 (0.35) CHRM5CHRM1CYP3A4POLBMAPT
SCHEMBL64456 0.75 PPARG (0.39) CHRM5CHRM1
SCHEMBL65299 0.75 LTA4H (0.35) CYP3A4KCNH2HRH3ESR1ESR2
SCHEMBL66854 0.74 CHRM2 (0.38) CHRM5CHRM1POLBTP53L3MBTL1
SCHEMBL78724 0.72 KDM4E (0.34) CHRM5CHRM1MAPTL3MBTL1
SCHEMBL91270 0.71 PPARG (0.38) CHRM5CHRM1POLBTP53L3MBTL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8129538-B1 Renin inhibitors TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2012-03-06 US disclosed