SCHEMBL6426783

SCHEMBL6426783

O=C1C(c2ccncc2)=C(C(F)(F)F)C(=O)N1Cc1ccccc1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NR1H2 P55055 3/20 0.47
NR1H3 Q13133 3/20 0.47
MAPK1 P28482 2/20 0.41
MAPT P10636 1/20 0.41
TDP1 Q9NUW8 1/20 0.41
CASP3 P42574 1/20 0.40
F2 P00734 1/20 0.40
PLG P00747 1/20 0.40
ELANE P08246 1/20 0.40
CTSG P08311 1/20 0.40
CMA1 P23946 1/20 0.40
CTRC Q99895 1/20 0.40
ALDH1A1 P00352 2/20 0.40
CHRM5 P08912 2/20 0.39
SIRT2 Q8IXJ6 1/20 0.39
P2RX7 Q99572 1/20 0.39
PKN1 Q16512 1/20 0.39
PKN2 Q16513 1/20 0.39
NPSR1 Q6W5P4 1/20 0.38
GSK3A P49840 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6427487 0.86 DHPS (0.46) NR1H2NR1H3ALDH1A1CHRM5KDM4E
SCHEMBL6428548 0.85 NR1H2 (0.56) NR1H2NR1H3MAPK1MAPTCASP3
SCHEMBL6428246 0.82 GSK3B (0.39) NR1H2NR1H3MAPK1MAPTTDP1
SCHEMBL6431729 0.80 NR1H2 (0.51) NR1H2NR1H3MAPK1MAPTTDP1
SCHEMBL6429546 0.80 OPRK1 (0.40) NR1H2NR1H3CASP3F2PLG
SCHEMBL6429024 0.80 PTGS2 (0.46) NR1H2NR1H3
SCHEMBL6427166 0.80 CASP1 (0.47) NR1H2NR1H3MAPTCASP3ALDH1A1
SCHEMBL6427122 0.77 NR1H2 (0.47) NR1H2NR1H3MAPTALDH1A1CHRM5
SCHEMBL6429398 0.76 NPSR1 (0.41) NR1H2NR1H3MAPK1MAPTCASP3
SCHEMBL6427820 0.75 KMT2A (0.47) NR1H2NR1H3MAPK1MAPTALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2005024755-A2 MEDICAMENTS FOR THE TREATMENT OF NEURODEGENERATIVE DISORDERS OR DIABETES DECIPHERA PHARMACEUTICALS, LLC. (US) 2005-03-17 WO disclosed