SCHEMBL6427487

SCHEMBL6427487

O=C1C(c2cccnc2)=C(C(F)(F)F)C(=O)N1Cc1ccccc1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
DHPS P49366 4/20 0.46
CYP2E1 P05181 1/20 0.45
CYP3A4 P08684 1/20 0.45
CYP2D6 P10635 1/20 0.45
CYP2A6 P11509 1/20 0.45
CYP2C9 P11712 1/20 0.45
CYP2B6 P20813 1/20 0.45
CYP2C19 P33261 1/20 0.45
L3MBTL1 Q9Y468 2/20 0.44
NR1H2 P55055 2/20 0.44
NR1H3 Q13133 2/20 0.44
CHRM5 P08912 1/20 0.43
KDM4E B2RXH2 1/20 0.42
UBE2N P61088 1/20 0.42
ATM Q13315 1/20 0.42
LMNA P02545 1/20 0.42
GAA P10253 1/20 0.41
ALDH1A1 P00352 1/20 0.41
SMN1; SMN2 Q16637 1/20 0.41
CCR9 P51686 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6426783 0.86 NR1H2 (0.47) NR1H2NR1H3CHRM5KDM4EALDH1A1
SCHEMBL6466541 0.82 L3MBTL1 (0.51) DHPSCYP2E1CYP3A4CYP2D6CYP2A6
SCHEMBL6428548 0.79 NR1H2 (0.56) L3MBTL1NR1H2NR1H3LMNAALDH1A1
SCHEMBL6429546 0.77 OPRK1 (0.40) CYP2C19NR1H2NR1H3ALDH1A1
SCHEMBL6428246 0.77 GSK3B (0.39) CYP2D6NR1H2NR1H3KDM4EALDH1A1
SCHEMBL4688137 0.75 KDM4E (0.51) DHPSCYP2E1CYP3A4CYP2D6CYP2A6
SCHEMBL6429024 0.74 PTGS2 (0.46) NR1H2NR1H3
SCHEMBL6427166 0.74 CASP1 (0.47) CYP2C19NR1H2NR1H3KDM4ELMNA
SCHEMBL6429398 0.73 NPSR1 (0.41) L3MBTL1NR1H2NR1H3ATMLMNA
SCHEMBL6427122 0.72 NR1H2 (0.47) NR1H2NR1H3CHRM5LMNAALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2005024755-A2 MEDICAMENTS FOR THE TREATMENT OF NEURODEGENERATIVE DISORDERS OR DIABETES DECIPHERA PHARMACEUTICALS, LLC. (US) 2005-03-17 WO disclosed