SCHEMBL6430970

SCHEMBL6430970

CC(C)(S)CN1CCC(CCO)CC1

nearest known ligand 0.35

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
ACHE P22303 2/20 0.33
HRH3 Q9Y5N1 1/20 0.33
MMP3 P08254 1/20 0.33
MMP8 P22894 1/20 0.33
LTA4H P09960 1/20 0.32
TYMP P19971 2/20 0.32
OPRM1 P35372 2/20 0.32
OPRK1 P41145 2/20 0.32
BRD4 O60885 1/20 0.31
AKR1C3 P42330 1/20 0.30
TACR2 P21452 1/20 0.30
ESR2 Q92731 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17471183 0.84 CHRM4 (0.36) ACHEHRH3MMP3MMP8LTA4H
SCHEMBL22366364 0.77 DRD2 (0.41) ACHEMMP3MMP8OPRK1AKR1C3
SCHEMBL15846086 0.76 ACHE (0.36) ACHEHRH3MMP3MMP8LTA4H
SCHEMBL1840988 0.75 SMN1; SMN2 (0.45) ACHEHRH3TYMP
SCHEMBL6431447 0.74 CYP2D6 (0.33)
SCHEMBL24926136 0.74 HSD11B1 (0.35) HRH3
SCHEMBL5677281 0.74 ALDH1A1 (0.43) OPRM1OPRK1
SCHEMBL3865970 0.73 ACHE (0.32) ACHEHRH3
SCHEMBL6428945 0.73 TYMP (0.33) ACHETYMP
SCHEMBL1318049 0.73 SLC18A3 (0.46) ACHEHRH3LTA4HTYMPOPRK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1126838-A4 NITROSATED AND NITROSYLATED NONSTEROIDAL ANTIINFLAMMATORY COMPOUNDS, COMPOSITIONS AND METHODS OF USE NITROMED INC (US) 2005-02-16 EP disclosed
US-20030207919-A1 Nitrosated and nitrosylated nonsteroidal antiinflammatory compounds, compositions and methods of use NICOX S.A. (FR) 2003-11-06 US disclosed
US-6593347-B2 Especially a nitrosated and/or nitrosylated arylpropionic acid, arylacetic acid, enolic anilide or an oxicam NITROMED, INC. 2003-07-15 US disclosed
US-20020016322-A1 Nitrosated and nitrosylated nonsteroidal antiinflammatory compounds, compositons and methods of use NICOX S.A. (FR) 2002-02-07 US disclosed
US-6297260-B1 Nitrosated and nitrosylated nonsteroidal antiinflammatory compounds, compositions and methods of use NITROMED, INC. 2001-10-02 US disclosed
EP-1126838-A1 NITROSATED AND NITROSYLATED NONSTEROIDAL ANTIINFLAMMATORY COMPOUNDS, COMPOSITIONS AND METHODS OF USE Nitromed, Inc. (US) 2001-08-29 EP disclosed
WO-2000025776-A1 NITROSATED AND NITROSYLATED NONSTEROIDAL ANTIINFLAMMATORY COMPOUNDS, COMPOSITIONS AND METHODS OF USE NITROMED, INC. (US) 2000-05-11 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20020016322-A1 Nitrosated and nitrosylated nonsteroidal antiinflammatory compounds, compositons and methods of use NOS2, NOS3, NOS1 ACHE 188/4885HRH3 3883/4885MMP3 717/4885
US-20030207919-A1 Nitrosated and nitrosylated nonsteroidal antiinflammatory compounds, compositions and methods of use NOS2, NOS1, NOS3 ACHE 283/4885HRH3 3700/4885MMP3 1048/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.