Bromide

Bromide

SCHEMBL6440482

Br.Br.Oc1c(CBr)cc(Cl)cc1CBr

nearest known ligand 0.47

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

ACHEADRA1AADRA1BADRA1DADRA2AADRA2BADRA2CADRB1ADRB2ADRB3APH1AAPH1BCHRM2CHRM3EZH2GRIN2AHTR1AHTR1BHTR1DHTR1FHTR3ANCSTNP2RY12PSEN1PSEN2PSENENSIGMAR1SLC6A2SLC6A3SLC6A4

The experimentally established mechanism targets of Bromide. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR1A known ✓ P08908 1/20 0.33
ADRA2A known ✓ P08913 1/20 0.33
ADRA2B known ✓ P18089 1/20 0.33
ADRA2C known ✓ P18825 1/20 0.33
SLC6A2 known ✓ P23975 1/20 0.33
ADRA1A known ✓ P35348 1/20 0.33
SLC6A3 known ✓ Q01959 1/20 0.33
HIF1A Q16665 5/20 0.47
CYP2C9 P11712 3/20 0.47
CYP2C19 P33261 2/20 0.47
HSD17B10 Q99714 6/20 0.42
CYP3A4 P08684 5/20 0.42
ALDH1A1 P00352 5/20 0.42
TSHR P16473 4/20 0.42
RECQL P46063 2/20 0.42
HPGD P15428 6/20 0.41
GABRA1 P14867 1/20 0.39
GABRB1 P18505 1/20 0.39
HSP90AA1 P07900 2/20 0.38
MEN1 O00255 4/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Bromide SCHEMBL6440480 1.00 HIF1A (0.47) HIF1ACYP2C9CYP2C19HSD17B10CYP3A4
SCHEMBL29516784 0.97 HIF1A (0.48) HIF1ACYP2C9CYP2C19HSD17B10CYP3A4
SCHEMBL9993152 0.86 HSD17B10 (0.56) HIF1ACYP2C9CYP2C19HSD17B10CYP3A4
SCHEMBL11591823 0.84 ERN1 (0.47) HIF1ACYP2C9CYP2C19HSD17B10CYP3A4
SCHEMBL29087535 0.78 HSPA5 (0.46) HIF1ACYP2C9CYP2C19HSD17B10CYP3A4
SCHEMBL21437010 0.76 BACE1 (0.39) ALDH1A1GABRA1ESR1ESR2
SCHEMBL1004123 0.74 CYP2C9 (0.50) HIF1ACYP2C9CYP2C19HSD17B10CYP3A4
SCHEMBL22543122 0.74 TRPA1 (0.33) CYP2C9HSD17B10ALDH1A1TSHRGABRA1
SCHEMBL11336884 0.74 HIF1A (0.50) HIF1ACYP2C9CYP2C19HSD17B10CYP3A4
SCHEMBL6443715 0.72 AMY1A (0.48) HIF1ACYP2C9CYP2C19HSD17B10ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6919456-B2 Catalytic compositions and methods for asymmetric aldol reactions THE BOARD OF TRUSTEES OF THE LELAND STANFORD JUNIOR UNIVERSITY (US) 2005-07-19 US disclosed
EP-1409122-A2 CATALYTIC COMPOSITIONS AND METHODS FOR ASYMMETRIC ALDOL REACTIONS THE BOARD OF TRUSTEES OF THE LELAND STANFORD JUNIOR UNIVERSITY (US) 2004-04-21 EP disclosed
US-20040019239-A1 Catalytic compositions and methods for asymmetric aldol reactions NATIONAL INSTITUTES OF HEALTH (NIH), U.S. DEPT. OF HEALTH AND HUMAN SERVICES (DHHS), U.S. GOVERNMENT 2004-01-29 US disclosed
US-6610889-B2 Using organometallic complex catalyst THE BOARD OF TRUSTEES OF THE LELAND STANFORD JUNIOR UNIVERSITY 2003-08-26 US disclosed
US-20020147367-A1 Catalytic compositions and methods for asymmetric aldol reactions NATIONAL INSTITUTES OF HEALTH (NIH), U.S. DEPT. OF HEALTH AND HUMAN SERVICES (DHHS), U.S. GOVERNMENT 2002-10-10 US disclosed
WO-2002041984-A2 CATALYTIC COMPOSITIONS AND METHODS FOR ASYMMETRIC ALDOL REACTIONS THE BOARD OF TRUSTEES OF THE LELAND STANFORD JUNIOR UNIVERSITY (US) 2002-05-30 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20020147367-A1 Catalytic compositions and methods for asymmetric aldol reactions ADH1C, ADH5, ADH1A HTR1A 3763/4885ADRA2A 739/4885ADRA2B 637/4885
US-20040019239-A1 Catalytic compositions and methods for asymmetric aldol reactions ADH1C, ADH5, ADH1A HTR1A 3763/4885ADRA2A 739/4885ADRA2B 637/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.