SCHEMBL6442508

SCHEMBL6442508

N#CCCNC(=O)C(C(N)=O)c1ccc(O)cc1

nearest known ligand 0.42

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
CNR1 P21554 1/20 0.40
CNR2 P34972 1/20 0.40
ESR1 P03372 7/20 0.36
ESR2 Q92731 7/20 0.36
CTSL P07711 1/20 0.34
MEN1 O00255 1/20 0.34
ALDH1A1 P00352 1/20 0.34
CYP1A2 P05177 1/20 0.34
CYP3A4 P08684 1/20 0.34
CYP2C9 P11712 1/20 0.34
CYP2C19 P33261 1/20 0.34
KMT2A Q03164 1/20 0.34
CTSS P25774 2/20 0.33
CTSK P43235 2/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6446778 0.87 CNR1 (0.43) CNR1CNR2CTSLCTSSCTSK
SCHEMBL6444717 0.85 CTSL (0.47) CNR1CNR2CTSLCTSSCTSK
SCHEMBL6445401 0.80 TNF (0.38) CTSLCYP3A4CTSSCTSK
SCHEMBL6020910 0.75 SLC7A5 (0.51)
SCHEMBL6446763 0.73 ESR1 (0.41) CNR1CNR2ESR1ESR2CTSL
SCHEMBL6443579 0.72 CTSS (0.38) CNR1CNR2ESR1ESR2CTSL
SCHEMBL6446787 0.72 CTSS (0.52) CTSLCTSSCTSK
SCHEMBL6825007 0.72 KDM4E (0.47) CNR1CNR2CTSLMEN1ALDH1A1
SCHEMBL6822727 0.71 CYP1A1 (0.40) CNR1CNR2ESR1ESR2CTSL
SCHEMBL6442609 0.71 CTSS (0.37) CNR1CNR2ESR1ESR2CTSL

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1575903-A1 COMPOUNDS FOR THE INHIBITION OF ROTAMASES Jerini AG (DE) 2005-09-21 EP claimed
WO-2004065353-A1 COMPOUNDS FOR THE INHIBITION OF ROTAMASES JERINI AG (DE) 2004-08-05 WO claimed
WO-2004056755-A2 COMPOUNDS FOR THE INHIBITION OF NON-PROTEOLYTIC ENZYMES JERENI AG (DE) 2004-07-08 WO claimed
EP-1575903-A1 COMPOUNDS FOR THE INHIBITION OF ROTAMASES Jerini AG (DE) 2005-09-21 EP disclosed
WO-2004065353-A1 COMPOUNDS FOR THE INHIBITION OF ROTAMASES JERINI AG (DE) 2004-08-05 WO disclosed
WO-2004056755-A2 COMPOUNDS FOR THE INHIBITION OF NON-PROTEOLYTIC ENZYMES JERENI AG (DE) 2004-07-08 WO disclosed