SCHEMBL6445401

SCHEMBL6445401

N#CCCNC(=O)C(C(N)=O)c1ccc2ccccc2c1

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TNF P01375 1/20 0.38
MTNR1A P48039 1/20 0.37
MTNR1B P49286 1/20 0.37
CTSS P25774 4/20 0.37
CTSB P07858 3/20 0.37
CTSL P07711 2/20 0.37
CTSK P43235 2/20 0.37
ATM Q13315 1/20 0.37
CYP3A4 P08684 2/20 0.37
CYP2D6 P10635 2/20 0.37
SLC6A2 P23975 2/20 0.37
SLC6A4 P31645 2/20 0.37
SLC6A3 Q01959 2/20 0.37
KCNH2 Q12809 1/20 0.37
MMP9 P14780 1/20 0.36
MC4R P32245 1/20 0.36
MC3R P41968 1/20 0.36
MC1R Q01726 1/20 0.36
HDAC1 Q13547 1/20 0.36
HDAC8 Q9BY41 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6446425 0.87 CTSS (0.48) MTNR1AMTNR1BCTSSCTSBCTSL
SCHEMBL6446778 0.84 CNR1 (0.43) CTSSCTSBCTSLCTSKEPHX1
SCHEMBL6442508 0.80 CNR1 (0.40) CTSSCTSLCTSKCYP3A4
SCHEMBL6447322 0.76 CTSK (0.42) CTSSCTSBCTSLCTSKATM
SCHEMBL6447648 0.76 MTNR1A (0.40) MTNR1AMTNR1BCTSSCTSBCTSL
SCHEMBL6020723 0.76 NLN (0.52) CTSSCTSBCTSLCTSK
SCHEMBL6443504 0.76 CTSK (0.37) MTNR1AMTNR1BCTSSCTSBCTSL
SCHEMBL5716820 0.75 UGT2B7 (0.53) TNFATMCYP3A4CYP2D6SLC6A2
SCHEMBL6573647 0.75 UGT2B7 (0.47) CYP3A4CYP2D6SLC6A2SLC6A4SLC6A3
SCHEMBL6575278 0.75 UGT2B7 (0.47) CYP3A4CYP2D6SLC6A2SLC6A4SLC6A3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1575903-A1 COMPOUNDS FOR THE INHIBITION OF ROTAMASES Jerini AG (DE) 2005-09-21 EP claimed
WO-2004065353-A1 COMPOUNDS FOR THE INHIBITION OF ROTAMASES JERINI AG (DE) 2004-08-05 WO claimed
WO-2004056755-A2 COMPOUNDS FOR THE INHIBITION OF NON-PROTEOLYTIC ENZYMES JERENI AG (DE) 2004-07-08 WO claimed
EP-1575903-A1 COMPOUNDS FOR THE INHIBITION OF ROTAMASES Jerini AG (DE) 2005-09-21 EP disclosed
WO-2004065353-A1 COMPOUNDS FOR THE INHIBITION OF ROTAMASES JERINI AG (DE) 2004-08-05 WO disclosed
WO-2004056755-A2 COMPOUNDS FOR THE INHIBITION OF NON-PROTEOLYTIC ENZYMES JERENI AG (DE) 2004-07-08 WO disclosed