SCHEMBL6446787

SCHEMBL6446787

N#CCNC(=O)C(C(N)=O)c1ccccc1

nearest known ligand 0.52

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
CTSS P25774 13/20 0.52
CTSL P07711 11/20 0.52
CTSB P07858 8/20 0.52
CTSK P43235 8/20 0.51
CTSC P53634 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6444717 0.87 CTSL (0.47) CTSSCTSLCTSBCTSKCTSC
SCHEMBL6446778 0.86 CNR1 (0.43) CTSSCTSLCTSBCTSK
SCHEMBL6446425 0.84 CTSS (0.48) CTSSCTSLCTSBCTSK
SCHEMBL4243720 0.80 KMT2A (0.49)
SCHEMBL6264970 0.80 CTSS (0.57) CTSSCTSLCTSBCTSKCTSC
SCHEMBL17365565 0.79 CTSS (0.56) CTSSCTSLCTSBCTSK
SCHEMBL17365596 0.79 CTSS (0.56) CTSSCTSLCTSBCTSK
SCHEMBL7330779 0.78 CTSS (0.54) CTSSCTSLCTSBCTSK
SCHEMBL14861481 0.78 HDAC1 (0.56)
SCHEMBL7746674 0.78 NAAA (0.60)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1575903-A1 COMPOUNDS FOR THE INHIBITION OF ROTAMASES Jerini AG (DE) 2005-09-21 EP claimed
WO-2004065353-A1 COMPOUNDS FOR THE INHIBITION OF ROTAMASES JERINI AG (DE) 2004-08-05 WO claimed
WO-2004056755-A2 COMPOUNDS FOR THE INHIBITION OF NON-PROTEOLYTIC ENZYMES JERENI AG (DE) 2004-07-08 WO claimed
EP-1575903-A1 COMPOUNDS FOR THE INHIBITION OF ROTAMASES Jerini AG (DE) 2005-09-21 EP disclosed
WO-2004065353-A1 COMPOUNDS FOR THE INHIBITION OF ROTAMASES JERINI AG (DE) 2004-08-05 WO disclosed
WO-2004056755-A2 COMPOUNDS FOR THE INHIBITION OF NON-PROTEOLYTIC ENZYMES JERENI AG (DE) 2004-07-08 WO disclosed