SCHEMBL6445386

SCHEMBL6445386

N#CCCNC(=O)C(CNC(=O)C=CC(=O)O)c1ccccc1

nearest known ligand 0.51

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.44
TAAR1 Q96RJ0 4/20 0.44
CTSS P25774 2/20 0.43
CTSK P43235 2/20 0.43
LMNA P02545 1/20 0.43
CYP2D6 P10635 1/20 0.43
CYP2C19 P33261 1/20 0.43
POLB P06746 1/20 0.40
CTSL P07711 1/20 0.40
KDM4A O75164 1/20 0.39
KMT2A Q03164 3/20 0.39
GAA P10253 1/20 0.39
MEN1 O00255 2/20 0.38
KDM4E B2RXH2 1/20 0.38
CNR1 P21554 1/20 0.36
CNR2 P34972 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6446751 0.91 TDP2 (0.39) ALDH1A1TAAR1CTSSCTSKLMNA
SCHEMBL6822579 0.89 CTSK (0.54) ALDH1A1TAAR1CTSSCTSKLMNA
SCHEMBL6442447 0.88 ALDH1A1 (0.38) ALDH1A1TAAR1CTSSCTSKLMNA
SCHEMBL6443547 0.86 CTSK (0.43) CTSSCTSKCYP2C19POLBCTSL
SCHEMBL6443588 0.81 NPC1 (0.51) CTSSCTSKPOLBCTSLKDM4A
SCHEMBL6445366 0.80 CTSS (0.47) ALDH1A1CTSSCTSKPOLBCTSL
SCHEMBL6443393 0.79 CTSK (0.43) CTSSCTSKCYP2D6CYP2C19POLB
SCHEMBL6446467 0.79 CTSK (0.49) ALDH1A1CTSSCTSKLMNACYP2D6
SCHEMBL6448077 0.78 KDM4E (0.54) TAAR1CTSSCTSKLMNACYP2C19
SCHEMBL6447305 0.78 CTSS (0.43) CTSSCTSKLMNAPOLBCTSL

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1575903-A1 COMPOUNDS FOR THE INHIBITION OF ROTAMASES Jerini AG (DE) 2005-09-21 EP claimed
WO-2004065353-A1 COMPOUNDS FOR THE INHIBITION OF ROTAMASES JERINI AG (DE) 2004-08-05 WO claimed
WO-2004056755-A2 COMPOUNDS FOR THE INHIBITION OF NON-PROTEOLYTIC ENZYMES JERENI AG (DE) 2004-07-08 WO claimed
EP-1575903-A1 COMPOUNDS FOR THE INHIBITION OF ROTAMASES Jerini AG (DE) 2005-09-21 EP disclosed
WO-2004065353-A1 COMPOUNDS FOR THE INHIBITION OF ROTAMASES JERINI AG (DE) 2004-08-05 WO disclosed
WO-2004056755-A2 COMPOUNDS FOR THE INHIBITION OF NON-PROTEOLYTIC ENZYMES JERENI AG (DE) 2004-07-08 WO disclosed