SCHEMBL6446464

SCHEMBL6446464

CN(C#N)C(=O)N(CCc1ccc(O)cc1)C(=O)C=CC(=O)O

nearest known ligand 0.43

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
OPRM1 P35372 2/20 0.38
OPRD1 P41143 2/20 0.38
OPRK1 P41145 2/20 0.38
ESRRG P62508 1/20 0.36
KDM4E B2RXH2 1/20 0.36
ALDH1A1 P00352 1/20 0.35
MAPT P10636 1/20 0.35
KMT2A Q03164 1/20 0.35
ATG4B Q9Y4P1 8/20 0.34
PLA2G1B P04054 7/20 0.34
LTB4R Q15722 2/20 0.34
LTB4R2 Q9NPC1 2/20 0.34
GLI1 P08151 1/20 0.34
GLI2 P10070 1/20 0.34
THRA P10827 1/20 0.33
THRB P10828 1/20 0.33
CYP1A2 P05177 1/20 0.33
TDP1 Q9NUW8 1/20 0.33
RECQL P46063 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6446460 1.00 OPRM1 (0.38) OPRM1OPRD1OPRK1ESRRGKDM4E
SCHEMBL6822577 0.90 LTB4R (0.43) ALDH1A1MAPTKMT2ALTB4RLTB4R2
SCHEMBL6822576 0.90 LTB4R (0.43) ALDH1A1MAPTKMT2ALTB4RLTB4R2
SCHEMBL6446747 0.85 ATG4B (0.35) OPRM1OPRD1OPRK1ALDH1A1MAPT
SCHEMBL6446750 0.85 ATG4B (0.35) OPRM1OPRD1OPRK1ALDH1A1MAPT
SCHEMBL6443833 0.82 SIGMAR1 (0.41) LTB4RLTB4R2CYP1A2
SCHEMBL6443830 0.82 SIGMAR1 (0.41) LTB4RLTB4R2CYP1A2
SCHEMBL6446222 0.76 ZDHHC20 (0.37) KMT2A
SCHEMBL6446217 0.76 ZDHHC20 (0.37) KMT2A
SCHEMBL6445379 0.75 ALDH1A1 (0.39) ALDH1A1MAPTKMT2ALTB4RLTB4R2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1575903-A1 COMPOUNDS FOR THE INHIBITION OF ROTAMASES Jerini AG (DE) 2005-09-21 EP claimed
WO-2004065353-A1 COMPOUNDS FOR THE INHIBITION OF ROTAMASES JERINI AG (DE) 2004-08-05 WO claimed
WO-2004056755-A2 COMPOUNDS FOR THE INHIBITION OF NON-PROTEOLYTIC ENZYMES JERENI AG (DE) 2004-07-08 WO claimed