SCHEMBL6444049

SCHEMBL6444049

CC(C)(C)OC(=O)NCC(C(=O)NCCC#N)c1ccc2ccccc2c1

nearest known ligand 0.50

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
CTSS P25774 16/20 0.50
CTSK P43235 13/20 0.50
CTSB P07858 6/20 0.50
CTSL P07711 4/20 0.41
ACACB O00763 1/20 0.39
GABRB1 P18505 1/20 0.39
GABRB2 P47870 1/20 0.39
KDM4A O75164 1/20 0.39
NQO2 P16083 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6445274 0.91 CTSS (0.60) CTSSCTSKCTSBCTSL
SCHEMBL6447648 0.89 MTNR1A (0.40) CTSSCTSKCTSBCTSL
SCHEMBL6445439 0.87 CTSS (0.56) CTSSCTSKCTSBCTSL
SCHEMBL6443381 0.87 CYP2D6 (0.40) CTSSCTSKCTSBCTSL
SCHEMBL6446829 0.85 CTSS (0.38) CTSSCTSKCTSBCTSL
SCHEMBL6443928 0.85 CTSK (0.41) CTSSCTSKCTSBCTSL
SCHEMBL6819019 0.84 CTSS (0.48) CTSSCTSKCTSBCTSLNQO2
SCHEMBL6575223 0.84 CTSS (0.46) CTSSCTSKCTSBACACBGABRB1
SCHEMBL6445255 0.83 NPC1 (0.44) CTSSCTSKCTSBCTSL
SCHEMBL6165666 0.83 CTSS (0.44) CTSSCTSKCTSBACACBGABRB1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1575903-A1 COMPOUNDS FOR THE INHIBITION OF ROTAMASES Jerini AG (DE) 2005-09-21 EP claimed
WO-2004065353-A1 COMPOUNDS FOR THE INHIBITION OF ROTAMASES JERINI AG (DE) 2004-08-05 WO claimed
WO-2004056755-A2 COMPOUNDS FOR THE INHIBITION OF NON-PROTEOLYTIC ENZYMES JERENI AG (DE) 2004-07-08 WO claimed
EP-1575903-A1 COMPOUNDS FOR THE INHIBITION OF ROTAMASES Jerini AG (DE) 2005-09-21 EP disclosed
WO-2004065353-A1 COMPOUNDS FOR THE INHIBITION OF ROTAMASES JERINI AG (DE) 2004-08-05 WO disclosed
WO-2004056755-A2 COMPOUNDS FOR THE INHIBITION OF NON-PROTEOLYTIC ENZYMES JERENI AG (DE) 2004-07-08 WO disclosed