SCHEMBL6462625

SCHEMBL6462625

CC(C)=C1Oc2cccc(OCCCN3CCC(NC(=O)Cc4ccccc4)CC3)c2C1=O

nearest known ligand 0.52

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
SIGMAR1 Q99720 5/20 0.52
CHRM1 P11229 12/20 0.51
CHRM2 P08172 1/20 0.51
CHRM4 P08173 1/20 0.51
CHRM5 P08912 1/20 0.51
DRD2 P14416 1/20 0.51
CHRM3 P20309 1/20 0.51
HTR2A P28223 1/20 0.51
ADRA1A P35348 1/20 0.51
HRH1 P35367 1/20 0.51
ADRA1B P35368 1/20 0.51
KCNH2 Q12809 1/20 0.51
MCHR1 Q99705 1/20 0.51
CCR8 P51685 2/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6458570 0.90 POLB (0.49) CHRM1CHRM2CHRM4CHRM5DRD2
SCHEMBL6457124 0.89 ADRA1D (0.50) DRD2HTR2AADRA1AHRH1ADRA1B
SCHEMBL6426288 0.87 CNR2 (0.48) CHRM1DRD2HTR2A
SCHEMBL6465555 0.85 SIGMAR1 (0.51) SIGMAR1ADRA1AADRA1B
SCHEMBL6462987 0.84 HTR7 (0.47) ADRA1AHRH1ADRA1B
SCHEMBL6466592 0.84 HTR7 (0.55) SIGMAR1DRD2HTR2AADRA1AHRH1
SCHEMBL6465657 0.83 HTR7 (0.57) DRD2ADRA1AADRA1B
SCHEMBL6461236 0.83 HTR7 (0.46) CHRM1ADRA1AHRH1ADRA1B
SCHEMBL6470095 0.83 EPHX2 (0.40) SIGMAR1DRD2HTR2A
SCHEMBL6472358 0.83 DRD4 (0.56) DRD2MCHR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1012147-B1 O-SUBSTITUTED HYDROXYCUMARANONE DERIVATIVES AS ANTITUMOR AND ANTIMETASTATIC AGENTS HOFFMANN LA ROCHE (CH) 2005-11-02 EP disclosed
US-6200989-B1 ADMINISTERING AS UROKINASE PLASMINOGEN ACTIVATOR ANTAGONISTS, ANTITUMOR AND ANTIMETASTASIS AGENTS HOFFMANN-LA ROCHE INC. 2001-03-13 US disclosed