SCHEMBL6465555

SCHEMBL6465555

CC(C)=C1Oc2cccc(OCCCN3CCC(NC(=O)Cc4c[nH]c5ccccc45)CC3)c2C1=O

nearest known ligand 0.51

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
SIGMAR1 Q99720 3/20 0.51
ADRA2A P08913 1/20 0.44
ADRA2B P18089 1/20 0.44
ADRA2C P18825 1/20 0.44
ADRA1D P25100 1/20 0.44
ADRA1A P35348 1/20 0.44
ADRA1B P35368 1/20 0.44
BCHE P06276 2/20 0.43
ACHE P22303 2/20 0.43
NPY5R Q15761 1/20 0.42
SOS1 Q07889 3/20 0.41
KRAS P01116 1/20 0.41
HPGD P15428 1/20 0.40
HTT P42858 1/20 0.40
RECQL P46063 1/20 0.40
HTR4 Q13639 3/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6462625 0.85 SIGMAR1 (0.52) SIGMAR1ADRA1AADRA1B
SCHEMBL6458570 0.82 POLB (0.49) ADRA1AADRA1B
SCHEMBL6457124 0.81 ADRA1D (0.50) ADRA1DADRA1AADRA1B
SCHEMBL6426288 0.81 CNR2 (0.48)
SCHEMBL6462987 0.78 HTR7 (0.47) ADRA1DADRA1AADRA1B
SCHEMBL6466592 0.78 HTR7 (0.55) SIGMAR1ADRA1DADRA1AADRA1B
SCHEMBL6461236 0.78 HTR7 (0.46) ADRA1DADRA1AADRA1B
SCHEMBL6465657 0.78 HTR7 (0.57) ADRA1DADRA1AADRA1BHPGD
SCHEMBL6470095 0.78 EPHX2 (0.40) SIGMAR1
SCHEMBL6472358 0.77 DRD4 (0.56)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1012147-B1 O-SUBSTITUTED HYDROXYCUMARANONE DERIVATIVES AS ANTITUMOR AND ANTIMETASTATIC AGENTS HOFFMANN LA ROCHE (CH) 2005-11-02 EP disclosed
US-6200989-B1 ADMINISTERING AS UROKINASE PLASMINOGEN ACTIVATOR ANTAGONISTS, ANTITUMOR AND ANTIMETASTASIS AGENTS HOFFMANN-LA ROCHE INC. 2001-03-13 US disclosed