SCHEMBL6470095

SCHEMBL6470095

CC(C)=C1Oc2cccc(OCCCN3CCC(NC4CCCCC4)CC3)c2C1=O

nearest known ligand 0.40

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
EPHX2 P34913 5/20 0.40
MAPT P10636 1/20 0.39
HTR1A P08908 5/20 0.38
HTR7 P34969 5/20 0.38
DRD2 P14416 1/20 0.38
HTR2A P28223 1/20 0.38
HTR6 P50406 1/20 0.38
BRD4 O60885 1/20 0.38
BRD2 P25440 1/20 0.38
BRD3 Q15059 1/20 0.38
ALDH1A1 P00352 3/20 0.37
KDM4E B2RXH2 2/20 0.37
MEN1 O00255 1/20 0.37
PKM P14618 1/20 0.37
KMT2A Q03164 1/20 0.37
S1PR5 Q9H228 1/20 0.37
SIGMAR1 Q99720 1/20 0.37
HRH3 Q9Y5N1 2/20 0.36
SMN1; SMN2 Q16637 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6457124 0.84 ADRA1D (0.50) HTR1AHTR7DRD2HTR2A
SCHEMBL6462625 0.83 SIGMAR1 (0.52) DRD2HTR2ASIGMAR1
SCHEMBL6466592 0.83 HTR7 (0.55) HTR1AHTR7DRD2HTR2AHTR6
SCHEMBL6462987 0.83 HTR7 (0.47) HTR1AHTR7ALDH1A1SMN1; SMN2
SCHEMBL6426288 0.82 CNR2 (0.48) DRD2HTR2AS1PR5
SCHEMBL6465657 0.82 HTR7 (0.57) HTR7DRD2ALDH1A1MEN1KMT2A
SCHEMBL6461236 0.82 HTR7 (0.46) HTR1AHTR7
SCHEMBL6458570 0.82 POLB (0.49) DRD2HTR2AHRH3
SCHEMBL6451907 0.82 POLB (0.50) HTR1AHTR7ALDH1A1
SCHEMBL6421954 0.81 ALDH1A1 (0.41) EPHX2MAPTALDH1A1KDM4EMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1012147-B1 O-SUBSTITUTED HYDROXYCUMARANONE DERIVATIVES AS ANTITUMOR AND ANTIMETASTATIC AGENTS HOFFMANN LA ROCHE (CH) 2005-11-02 EP disclosed
EP-1012147-A2 O-SUBSTITUTED HYDROXYCUMARANONE DERIVATIVES AS ANTITUMOR AND ANTIMETASTATIC AGENTS F. HOFFMANN-LA ROCHE AG (CH) 2000-06-28 EP disclosed
WO-1999006387-A2 O-SUBSTITUTED HYDROXYCUMARANONE DERIVATIVES AS ANTITUMOR AND ANTIMETASTATIC AGENTS F. HOFFMANN-LA ROCHE AG (CH) 1999-02-11 WO disclosed