SCHEMBL6464905

SCHEMBL6464905

Nc1nc2[nH]cnc2c(=O)n1C[C]=O

nearest known ligand 0.35

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
PNP P00491 2/20 0.35
ADORA2B P29275 6/20 0.34
ADORA3 P0DMS8 2/20 0.34
ADORA2A P29274 6/20 0.32
PDE4A P27815 5/20 0.32
PDE4B Q07343 5/20 0.32
PDE4C Q08493 5/20 0.32
PDE4D Q08499 5/20 0.32
LMNA P02545 1/20 0.30
CYP1A2 P05177 1/20 0.30
MAPT P10636 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6267115 0.87 ADORA2B (0.48) PNPADORA2BADORA3ADORA2APDE4A
SCHEMBL9960806 0.84 PNP (0.38) PNPADORA2BADORA3ADORA2APDE4A
SCHEMBL874734 0.82 ADORA2A (0.45) PNPADORA2BADORA3ADORA2APDE4A
SCHEMBL669004 0.79 ADORA2B (0.50) PNPADORA2BADORA3ADORA2APDE4A
SCHEMBL3671337 0.79 PNP (0.37) PNPADORA2BADORA3ADORA2APDE4A
SCHEMBL667794 0.79 PDE4A (0.49) ADORA2BADORA3ADORA2APDE4APDE4B
SCHEMBL5048171 0.78 PNP (0.39) PNPADORA2BPDE4APDE4BPDE4C
SCHEMBL5503490 0.78 ADORA2A (0.49) PNPADORA2BADORA3ADORA2APDE4A
SCHEMBL17186375 0.78 KDM5B (0.39) PNP
SCHEMBL21748352 0.78 ADORA2A (0.40) PNPADORA2BADORA2ALMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-11839661-B2 Rapid formation of supramolecular hydrogels by short peptide and bioactive small molecules BRANDEIS UNIVERSITY (US) 2023-12-12 US disclosed
US-20210128745-A1 RAPID FORMATION OF SUPRAMOLECULAR HYDROGELS BY SHORT PEPTIDE AND BIOACTIVE SMALL MOLECULES BRANDEIS UNIVERSITY 2021-05-06 US disclosed
WO-2019035928-A1 RAPID FORMATION OF SUPRAMOLECULAR HYDROGELS BY SHORT PEPTIDE AND BIOACTIVE SMALL MOLECULES BRANDEIS UNIVERSITY (US) 2019-02-21 WO disclosed
US-8188011-B1 Optimization of ligand affinity for RNA targets using mass spectrometry ISIS PHARMACEUTICALS, INC. (US) 2012-05-29 US disclosed
US-20050142581-A1 Microrna as ligands and target molecules ISIS PHARMACEUTICALS, INC. 2005-06-30 US disclosed
US-6849660-B1 Antimicrobial biaryl compounds ISIS PHARMACEUTICALS, INC. (US) 2005-02-01 US disclosed
US-6770486-B1 IDENTIFICATION OF LIGAND COMPOUNDS THAT BIND TO TARGET MOLECULES SUCH AS PROTEINS OR STRUCTURED RNA WITH AS LITTLE AS MILLIMOLAR (MM) AFFINITY USING MASS SPECTROMETRY ISIS PHARMACEUTICALS, INC. 2004-08-03 US disclosed