SCHEMBL6465769

SCHEMBL6465769

CC(C)CC(NC(=O)O)C(=O)NC(CCc1ccccc1)C(O)c1nc(C(=O)N2CCCc3ccccc32)co1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 5/20 0.39
MAPT P10636 4/20 0.39
RAB9A P51151 2/20 0.39
CTSS P25774 2/20 0.39
NPSR1 Q6W5P4 2/20 0.38
TSHR P16473 1/20 0.38
NPC1 O15118 1/20 0.37
LMNA P02545 1/20 0.37
SMN1; SMN2 Q16637 1/20 0.37
PSMB8 P28062 1/20 0.37
PSMB5 P28074 1/20 0.37
PSMB10 P40306 1/20 0.37
PSMB2 P49721 1/20 0.37
PDE4B Q07343 1/20 0.37
AVPR2 P30518 1/20 0.37
OXTR P30559 1/20 0.37
AVPR1A P37288 1/20 0.37
REN P00797 1/20 0.36
USP2 O75604 1/20 0.36
POLB P06746 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7042159 0.92 CTSK (0.45) CTSS
SCHEMBL6462350 0.87 CTSL (0.45) CTSS
SCHEMBL6466880 0.85 PSMB2 (0.45) MAPTCTSSPSMB8PSMB5PSMB10
SCHEMBL6465946 0.85 ALDH1A1 (0.41) ALDH1A1MAPTRAB9ACTSSNPSR1
SCHEMBL6466258 0.79 ANPEP (0.46) RAB9ANPC1SMN1; SMN2PSMB5PSMB2
SCHEMBL6467305 0.78 MMP9 (0.44) LMNAPSMB5PSMB2REN
SCHEMBL6467310 0.78 MMP9 (0.44) LMNAPSMB5PSMB2REN
SCHEMBL6466256 0.78 MMP9 (0.44) LMNAPSMB5PSMB2REN
SCHEMBL6061535 0.78 CTSK (0.51) CTSS
SCHEMBL6063162 0.78 CTSL (0.45) CTSS

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1516877-A1 Amine derivatives as protease inhibitors AXYS PHARMACEUTICALS, INC. (US) 2005-03-23 EP disclosed