Trolamine

Trolamine

SCHEMBL6479985

O=C(O)C=CC(=O)O.O=C(O)C=CC(=O)O.O=C(O)C=CC(=O)O.OCCN(CCO)CCO

nearest known ligand 0.50

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

ACEADRA1AADRA1BADRA1DADRA2AADRA2BADRA2CADRB1ADRB2ATP4AATP4BAXLBTKCACNA1CCACNA1DCACNA1FCACNA1SCCR5CHRM2CHRM3CPT1BCPT2DPP4DRD1DRD2EGFRERBB2ERBB4FLT3HRH1HRH3HTR1AHTR2AHTR2BHTR2CHTR4JAK1JAK2JAK3KCNH2KMT2AMAP2K1MAP2K2MEN1MLNRMPLMTORPPIK3CAPIK3CBPIK3CDPIK3CGPIK3R1PIK3R2PIK3R3PIK3R5PLK4PPARGRENS1PR1SLC6A2SLC6A3SLC6A4SMOTYK2atpAatpBatpCatpDatpEatpFatpFHatpGpol

The experimentally established mechanism targets of Trolamine. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MEN1 known ✓ O00255 1/20 0.34
KMT2A known ✓ Q03164 1/20 0.34
ACE known ✓ P12821 1/20 0.33
CHRM2 known ✓ P08172 1/20 0.32
ADRA2A known ✓ P08913 1/20 0.32
DRD1 known ✓ P21728 1/20 0.32
SLC6A2 known ✓ P23975 1/20 0.32
SLC6A4 known ✓ P31645 1/20 0.32
ADRA1A known ✓ P35348 1/20 0.32
SLC6A3 known ✓ Q01959 1/20 0.32
HRH3 known ✓ Q9Y5N1 1/20 0.32
TSHR P16473 5/20 0.50
TP53 P04637 1/20 0.50
EGLN1 Q9GZT9 1/20 0.50
EGLN3 Q9H6Z9 1/20 0.50
ALDH1A1 P00352 4/20 0.42
KDM4E B2RXH2 2/20 0.39
ALOX15 P16050 2/20 0.39
MAPT P10636 2/20 0.39
SMN1; SMN2 Q16637 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Trolamine SCHEMBL5874734 1.00 TSHR (0.50) TSHRTP53EGLN1EGLN3ALDH1A1
Trolamine SCHEMBL30358483 1.00 TSHR (0.50) TSHRTP53EGLN1EGLN3ALDH1A1
Trolamine SCHEMBL4944905 1.00 TSHR (0.50) TSHRTP53EGLN1EGLN3ALDH1A1
Trolamine SCHEMBL4944913 1.00 TSHR (0.50) TSHRTP53EGLN1EGLN3ALDH1A1
Trolamine SCHEMBL5875419 1.00 TSHR (0.50) TSHRTP53EGLN1EGLN3ALDH1A1
Trolamine SCHEMBL14989224 1.00 TSHR (0.50) TSHRTP53EGLN1EGLN3ALDH1A1
Trolamine SCHEMBL6838017 0.97 TSHR (0.47) TSHRTP53EGLN1EGLN3ALDH1A1
Trolamine SCHEMBL28088241 0.95 TSHR (0.45) TSHRTP53EGLN1EGLN3ALDH1A1
Trolamine SCHEMBL27950677 0.89 ALDH1A1 (0.41) TSHRTP53EGLN1EGLN3ALDH1A1
Fumaric Acid SCHEMBL1131856 0.85 ALDH1A1 (0.50) ALDH1A1HCAR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 11 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20050218517-A1 Semiconductor flip-chip package and method for the fabrication thereof M.A. CAPOTE (US) 2005-10-06 US disclosed
US-6774493-B2 INTEGRATED CIRCUIT COATED WITH THERMOSETTING POLYMER, WITH HARDENED ADHESIVE POLYMER UNDERFILL ENCAPSULANT INCLUDING INTERMIXED REACTION PRODUCT OF THERMOSETTING POLYMER AND FLUXING AGENT THAT CHEMICALLY IMMOBILIZES FLUX AND BY-PRODUCTS M. A. CAPOTE 2004-08-10 US disclosed
US-20030218261-A1 INTEGRATED CIRCUIT COATED WITH THERMOSETTING POLYMER, WITH HARDENED ADHESIVE POLYMER UNDERFILL ENCAPSULANT INCLUDING INTERMIXED REACTION PRODUCT OF THERMOSETTING POLYMER AND FLUXING AGENT THAT CHEMICALLY IMMOBILIZES FLUX AND BY-PRODUCTS M. A. CAPOTE (US) 2003-11-27 US disclosed
US-6566234-B1 Semiconductor flip-chip package and method for the fabrication thereof AGUILA TECHNOLOGIES, INC. 2003-05-20 US disclosed
US-6518677-B1 Semiconductor flip-chip package and method for the fabrication thereof Capote, Miguel Albert 2003-02-11 US disclosed
US-6132646-A ELECTROCONDUCTIVE INK AND CURING ADHESIVE WITH FLUX AND METALS MIGUEL ALBERT CAPOTE (US) 2000-10-17 US disclosed
EP-1025587-A4 SEMICONDUCTOR FLIP-CHIP PACKAGE AND METHOD FOR THE FABRICATION THEREOF AGUILA TECHNOLOGIES INC (US) 2000-10-04 EP disclosed
US-6121689-A Semiconductor flip-chip package and method for the fabrication thereof MIGUEL ALBERT CAPOTE (US) 2000-09-19 US disclosed
EP-1025587-A1 SEMICONDUCTOR FLIP-CHIP PACKAGE AND METHOD FOR THE FABRICATION THEREOF Aguila Technologies, Inc. (US) 2000-08-09 EP disclosed
US-5985043-A THERMALLY CURABLE ADHESIVE COMPRISING ACID HAVING TWO OR MORE DOUBLE BONDS AS FLUXING AGENT, DOUBLE BOND CONTAINING DILUENT CAPABLE OF CROSSLINKING FLUXING AGENT, OPTIONALLY FREE RADICAL INITIATOR, RESIN MIGUEL ALBERT CAPOTE (US) 1999-11-16 US disclosed
WO-1999004430-A1 SEMICONDUCTOR FLIP-CHIP PACKAGE AND METHOD FOR THE FABRICATION THEREOF AGUILA TECHNOLOGIES, INC. (US) 1999-01-28 WO disclosed