SCHEMBL6497035

SCHEMBL6497035

Cc1cccc(-c2ccc(C(F)(F)F)cc2)c1C(=O)O

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
BACE1 P56817 1/20 0.47
CYP2C8 P10632 1/20 0.46
DHODH Q02127 3/20 0.45
APP P05067 1/20 0.44
RXRA P19793 1/20 0.43
RXRB P28702 1/20 0.43
KIF11 P52732 1/20 0.43
PSEN1 P49768 1/20 0.42
PSEN2 P49810 1/20 0.42
APH1B Q8WW43 1/20 0.42
NCSTN Q92542 1/20 0.42
APH1A Q96BI3 1/20 0.42
PSENEN Q9NZ42 1/20 0.42
AKR1C3 P42330 1/20 0.42
AKR1C2 P52895 1/20 0.42
MEN1 O00255 1/20 0.41
MAPT P10636 1/20 0.41
HTT P42858 1/20 0.41
RAB9A P51151 1/20 0.41
KMT2A Q03164 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL593309 0.89 CYP2C8 (0.51) BACE1CYP2C8DHODHAPPRXRA
SCHEMBL7041867 0.84 BACE1 (0.44) BACE1MEN1MAPTHTTRAB9A
SCHEMBL30755410 0.84 BACE1 (0.44) BACE1MEN1MAPTHTTRAB9A
SCHEMBL23354520 0.83 RXRA (0.51) BACE1CYP2C8DHODHAPPRXRA
SCHEMBL31676846 0.83 RXRA (0.51) BACE1CYP2C8DHODHAPPRXRA
SCHEMBL23354270 0.83 IL2 (0.49) BACE1CYP2C8DHODHAPPKIF11
SCHEMBL22703438 0.82 TDP1 (0.46) DHODHAKR1C3MEN1RAB9AKMT2A
SCHEMBL27371068 0.81 APP (0.43) BACE1DHODHAPPRXRAMEN1
SCHEMBL29485413 0.81 FOLH1 (0.53) MEN1KMT2ATDP1L3MBTL1
SCHEMBL3229734 0.81 FOLH1 (0.53) MEN1KMT2ATDP1L3MBTL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8114993-B2 Use of aryl chlorides in palladium-catalyzed C-H bond functionalization THE UNIVERSITY OF HOUSTON SYSTEM (US) 2012-02-14 US disclosed
US-8114993-B2 Use of aryl chlorides in palladium-catalyzed C-H bond functionalization THE UNIVERSITY OF HOUSTON SYSTEM (US) 2012-02-14 US disclosed
US-20090012293-A1 USE OF ARYL CHLORIDES IN PALLADIUM-CATALYZED C-H BOND FUNCTIONALIZATION THE UNIVERSITY OF HOUSTON SYSTEM (US) 2009-01-08 US disclosed
US-20090012293-A1 USE OF ARYL CHLORIDES IN PALLADIUM-CATALYZED C-H BOND FUNCTIONALIZATION THE UNIVERSITY OF HOUSTON SYSTEM (US) 2009-01-08 US disclosed
US-20050038035-A1 Heterocyclic amide compounds as apolipoprotein b inhibitors DAISO CO., LTD. (JP) 2005-02-17 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20090012293-A1 USE OF ARYL CHLORIDES IN PALLADIUM-CATALYZED C-H BOND FUNCTIONALIZATION DBH, DDT, CYCS BACE1 4452/4885CYP2C8 77/4885DHODH 226/4885
US-20050038035-A1 Heterocyclic amide compounds as apolipoprotein b inhibitors APOB, APOL1, CTRB2 BACE1 49/4885CYP2C8 710/4885DHODH 4355/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.