SCHEMBL651079

SCHEMBL651079

CCCCn1c(-c2ccccc2C)nc(-c2ccc(C)cc2)c1CC(NCc1ccc(C(=O)O)cc1)C1CCCCC1

nearest known ligand 0.36

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
AGTR1 P30556 5/20 0.34
MME P08473 3/20 0.34
ADORA3 P0DMS8 1/20 0.34
ADORA2B P29275 1/20 0.34
ADORA1 P30542 1/20 0.34
PPARG P37231 1/20 0.33
MDM2 Q00987 1/20 0.33
AGTR2 P50052 1/20 0.33
LTB4R2 Q9NPC1 1/20 0.33
ALDH1A1 P00352 1/20 0.33
LMNA P02545 1/20 0.33
HPGD P15428 1/20 0.33
TDP1 Q9NUW8 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL653481 0.93 MERTK (0.34) AGTR1ADORA3ADORA2BALDH1A1LMNA
SCHEMBL648999 0.86 ADORA3 (0.37) AGTR1ADORA3ADORA2BADORA1PPARG
SCHEMBL651281 0.85 ADORA3 (0.37) AGTR1MMEADORA3ADORA2BADORA1
SCHEMBL650385 0.84 ADORA3 (0.36) AGTR1ADORA3ADORA2BADORA1PPARG
SCHEMBL650059 0.84 AGTR1 (0.37) AGTR1MMEADORA3ADORA2BADORA1
SCHEMBL652064 0.83 ITGB1 (0.31) ADORA3ADORA2B
SCHEMBL650087 0.83 ADORA3 (0.35) AGTR1ADORA3ADORA2BADORA1PPARG
SCHEMBL651088 0.79 LTB4R2 (0.40) AGTR1MMEPPARGLTB4R2
SCHEMBL652331 0.78 DRD2 (0.35) AGTR1ADORA2B
SCHEMBL4764000 0.78 ALDH1A1 (0.42) ADORA3ADORA2BADORA1ALDH1A1HPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8119665-B2 Aryl imidazoles and related compounds as C5a receptor modulators NOVARTIS INTERNATIONAL PHARMACEUTICAL LTD. (BM) 2012-02-21 US disclosed