SCHEMBL650318

SCHEMBL650318

C[C@H](NC(=O)c1cc2[nH]nc(NC(=O)c3ccccc3N)c2o1)c1ccccc1

nearest known ligand 0.55

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.55
KDM4E B2RXH2 1/20 0.55
MAPK1 P28482 15/20 0.48
BDKRB1 P46663 1/20 0.48
LMNA P02545 1/20 0.47
THRB P10828 1/20 0.47
AURKA O14965 2/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL653980 1.00 ALDH1A1 (0.55) ALDH1A1KDM4EMAPK1BDKRB1LMNA
SCHEMBL652872 0.85 BDKRB1 (0.45) ALDH1A1MAPK1BDKRB1LMNATHRB
SCHEMBL653508 0.85 BDKRB1 (0.45) ALDH1A1MAPK1BDKRB1LMNATHRB
SCHEMBL651126 0.85 NPC1 (0.41) ALDH1A1KDM4EBDKRB1LMNA
SCHEMBL652682 0.82 AURKA (0.53) MAPK1AURKA
SCHEMBL655164 0.81 AURKA (0.42) ALDH1A1KDM4EMAPK1BDKRB1AURKA
SCHEMBL653285 0.78 DYRK1A (0.41) ALDH1A1MAPK1
SCHEMBL653335 0.77 FADS1 (0.36) ALDH1A1KDM4EMAPK1AURKA
SCHEMBL2912045 0.74 CYP1A2 (0.42) ALDH1A1KDM4EMAPK1BDKRB1LMNA
SCHEMBL4290720 0.73 ALDH1A1 (1.00) ALDH1A1KDM4ELMNATHRB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8119641-B2 1H-furo[3,2-C]pyrazole compounds useful as kinase inhibitors NERVIANO MEDICAL SCIENCES S.R.L. (IT) 2012-02-21 US disclosed