SCHEMBL6504646

SCHEMBL6504646

O=C(Nc1nc2ccccc2n(CCN2CCOCC2)c1=O)c1ccccc1Cl

nearest known ligand 0.58

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HSD17B10 Q99714 4/20 0.58
CASP1 P29466 1/20 0.58
CASP7 P55210 1/20 0.58
L3MBTL1 Q9Y468 1/20 0.58
KDM4E B2RXH2 2/20 0.57
NPSR1 Q6W5P4 2/20 0.57
PYGM P11217 1/20 0.54
MAPK1 P28482 2/20 0.52
HPGD P15428 3/20 0.50
LMNA P02545 3/20 0.50
ALDH1A1 P00352 2/20 0.50
SMN1; SMN2 Q16637 2/20 0.50
KMT2A Q03164 2/20 0.50
MEN1 O00255 1/20 0.50
USP2 O75604 1/20 0.50
MAPT P10636 1/20 0.50
HTT P42858 1/20 0.50
TDP1 Q9NUW8 1/20 0.50
TSHR P16473 2/20 0.49
OPRK1 P41145 4/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6529548 0.87 HSD17B10 (0.54) HSD17B10CASP1CASP7L3MBTL1KDM4E
SCHEMBL6499836 0.87 KDM4E (0.74) HSD17B10CASP1CASP7L3MBTL1KDM4E
SCHEMBL6532182 0.86 KDM4E (0.77) HSD17B10CASP1CASP7L3MBTL1KDM4E
SCHEMBL6497804 0.86 KDM4E (0.64) HSD17B10CASP1CASP7L3MBTL1KDM4E
SCHEMBL6503393 0.84 HSD17B10 (0.62) HSD17B10CASP1CASP7L3MBTL1KDM4E
SCHEMBL6500237 0.84 KDM4E (0.62) HSD17B10CASP1CASP7L3MBTL1KDM4E
SCHEMBL6505494 0.78 HSD17B10 (0.58) HSD17B10CASP1CASP7L3MBTL1KDM4E
SCHEMBL5551592 0.77 LMNA (0.62) HSD17B10CASP1CASP7L3MBTL1KDM4E
SCHEMBL6529612 0.74 CASP1 (0.60) HSD17B10CASP1CASP7L3MBTL1KDM4E
SCHEMBL14470780 0.73 PYGM (0.69) HSD17B10CASP1CASP7L3MBTL1KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2005021547-A3 HETEROCYCLIC CANNABINOID CB2 RECEPTOR ANTAGONISTS PHARMAXIS PTY LTD (AU) 2005-08-18 WO disclosed
WO-2005021547-A2 HETEROCYCLIC CANNABINOID CB2 RECEPTOR ANTAGONISTS PHARMAXIS PTY LTD. (AU) 2005-03-10 WO disclosed