SCHEMBL6505494

SCHEMBL6505494

CC(C)(C)OC(=O)Nc1nc2ccccc2n(CCN2CCOCC2)c1=O

nearest known ligand 0.58

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HSD17B10 Q99714 2/20 0.58
CASP1 P29466 1/20 0.58
CASP7 P55210 1/20 0.58
L3MBTL1 Q9Y468 1/20 0.58
OPRM1 P35372 1/20 0.53
OPRD1 P41143 1/20 0.53
OGFRL1 Q5TC84 1/20 0.53
PYGM P11217 2/20 0.52
LMNA P02545 3/20 0.51
KDM4E B2RXH2 3/20 0.50
NPSR1 Q6W5P4 2/20 0.50
CNR2 P34972 1/20 0.46
GAA P10253 2/20 0.46
MAPT P10636 2/20 0.46
ALDH1A1 P00352 3/20 0.46
SMN1; SMN2 Q16637 2/20 0.46
CD274 Q9NZQ7 1/20 0.46
MTOR P42345 1/20 0.45
IRAK1 P51617 1/20 0.45
IRAK4 Q9NWZ3 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6503393 0.84 HSD17B10 (0.62) HSD17B10CASP1CASP7L3MBTL1PYGM
SCHEMBL8861171 0.84 OPRM1 (0.54) HSD17B10OPRM1OPRD1OGFRL1LMNA
SCHEMBL6497804 0.82 KDM4E (0.64) HSD17B10CASP1CASP7L3MBTL1OPRM1
SCHEMBL6504646 0.78 HSD17B10 (0.58) HSD17B10CASP1CASP7L3MBTL1OPRM1
SCHEMBL6532182 0.78 KDM4E (0.77) HSD17B10CASP1CASP7L3MBTL1OPRM1
SCHEMBL6529548 0.78 HSD17B10 (0.54) HSD17B10CASP1CASP7L3MBTL1PYGM
SCHEMBL14470780 0.77 PYGM (0.69) HSD17B10CASP1CASP7L3MBTL1PYGM
SCHEMBL6500237 0.76 KDM4E (0.62) HSD17B10CASP1CASP7L3MBTL1OPRM1
SCHEMBL6529612 0.74 CASP1 (0.60) HSD17B10CASP1CASP7L3MBTL1PYGM
SCHEMBL6529413 0.73 LMNA (0.58) HSD17B10CASP1CASP7L3MBTL1OPRM1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2005021547-A3 HETEROCYCLIC CANNABINOID CB2 RECEPTOR ANTAGONISTS PHARMAXIS PTY LTD (AU) 2005-08-18 WO disclosed
WO-2005021547-A2 HETEROCYCLIC CANNABINOID CB2 RECEPTOR ANTAGONISTS PHARMAXIS PTY LTD. (AU) 2005-03-10 WO disclosed
WO-2005021547-A2 HETEROCYCLIC CANNABINOID CB2 RECEPTOR ANTAGONISTS PHARMAXIS PTY LTD. (AU) 2005-03-10 WO disclosed