SCHEMBL6505249

SCHEMBL6505249

CCOc1cc(-c2ccc(F)cc2)ccc1C(=O)O

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADRB1 P08588 1/20 0.52
ADRB3 P13945 1/20 0.52
RARB P10826 3/20 0.50
RARA P10276 2/20 0.50
NEK2 P51955 1/20 0.47
MKNK1 Q9BUB5 1/20 0.47
MKNK2 Q9HBH9 1/20 0.47
HSD17B10 Q99714 2/20 0.46
TSHR P16473 1/20 0.46
MCL1 Q07820 1/20 0.46
CHRNA7 P36544 1/20 0.45
RXRA P19793 2/20 0.45
RXRB P28702 2/20 0.45
RXRG P48443 1/20 0.45
RARG P13631 1/20 0.45
KDM4E B2RXH2 2/20 0.44
SSTR5 P35346 2/20 0.44
CAMKK1 Q8N5S9 1/20 0.44
CAMKK2 Q96RR4 1/20 0.44
MEN1 O00255 2/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2769244 0.91 ADRB1 (0.55) ADRB1ADRB3RARBRARANEK2
SCHEMBL15630531 0.88 ADRB1 (0.55) ADRB1ADRB3RARBRARARARG
SCHEMBL4600863 0.88 PTPN11 (0.56) RARBRARAHSD17B10TSHRCHRNA7
SCHEMBL6498950 0.88 ADRB3 (0.60) ADRB1ADRB3NEK2MKNK1MKNK2
SCHEMBL15048810 0.87 TSHR (0.51) HSD17B10TSHRKDM4EMEN1KMT2A
SCHEMBL16616127 0.85 TDP1 (0.57) ADRB1ADRB3MKNK1MKNK2HSD17B10
SCHEMBL6496898 0.85 KDM4E (0.53) ADRB1ADRB3RARBRARANEK2
SCHEMBL3133634 0.83 ALDH1A1 (0.56) ADRB1ADRB3NEK2HSD17B10MCL1
SCHEMBL9518777 0.78 DCLRE1B (0.55) RARBRARAHSD17B10MCL1RARG
SCHEMBL1188345 0.78 TSHR (0.56) HSD17B10TSHRKDM4EMEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6884821-B1 Carboxylic acid derivatives and drugs containing the same EISAI CO., LTD. (JP) 2005-04-26 US disclosed
EP-1216980-A1 CARBOXYLIC ACID DERIVATIVES AND DRUGS CONTAINING THE SAME Eisai Co., Ltd. (JP) 2002-06-26 EP disclosed