SCHEMBL6505593

SCHEMBL6505593

Cc1sc(-c2ccccc2Cl)nc1C(=O)NCc1cc(CC(OC(C)C)C(=O)OC(=O)C(F)(F)F)ccn1

nearest known ligand 0.35

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADORA2A P29274 3/20 0.35
ADORA1 P30542 2/20 0.35
HPGD P15428 4/20 0.35
ALDH1A1 P00352 2/20 0.35
NPC1 O15118 1/20 0.35
CYP1A2 P05177 1/20 0.35
CYP3A4 P08684 1/20 0.35
CYP2C19 P33261 1/20 0.35
TSHR P16473 1/20 0.34
HTT P42858 1/20 0.34
PDE2A O00408 1/20 0.33
PIK3CD O00329 1/20 0.33
PPARD Q03181 1/20 0.33
PPARA Q07869 1/20 0.33
KDM4E B2RXH2 1/20 0.33
RAB9A P51151 1/20 0.33
VEGFA P15692 1/20 0.32
FLT1 P17948 1/20 0.32
EGLN1 Q9GZT9 1/20 0.32
EGLN3 Q9H6Z9 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6495822 0.92 SHMT1 (0.39) HPGDKDM4ECDC7DBF4
SCHEMBL6499174 0.90 ADORA1 (0.38) ADORA2AADORA1HPGDALDH1A1NPC1
SCHEMBL6531507 0.90 PARP1 (0.36) ADORA2AHPGDALDH1A1NPC1CYP1A2
Trifluoroacetic Acid SCHEMBL6505587 0.89 PPARA (0.38) ADORA2AADORA1HPGDALDH1A1NPC1
SCHEMBL6504395 0.89 PPARA (0.37) PPARDPPARA
SCHEMBL6505045 0.87 SMN1; SMN2 (0.35) ADORA2AADORA1HPGDALDH1A1NPC1
SCHEMBL6498709 0.87 CDK2 (0.34) NPC1PPARDPPARA
SCHEMBL6503597 0.86 KDM4E (0.36) ALDH1A1NPC1KDM4ERAB9APOLB
SCHEMBL6494741 0.85 PPARA (0.39) ADORA2AADORA1CYP1A2CYP3A4CYP2C19
Trifluoroacetic Acid SCHEMBL6495816 0.81 SHMT1 (0.44) PPARDPPARAKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6884821-B1 Carboxylic acid derivatives and drugs containing the same EISAI CO., LTD. (JP) 2005-04-26 US disclosed
EP-1216980-A1 CARBOXYLIC ACID DERIVATIVES AND DRUGS CONTAINING THE SAME Eisai Co., Ltd. (JP) 2002-06-26 EP disclosed