SCHEMBL6503597

SCHEMBL6503597

Cc1sc(-c2cccs2)nc1C(=O)NCc1cc(CC(OC(C)C)C(=O)OC(=O)C(F)(F)F)ccn1

nearest known ligand 0.36

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 10/20 0.36
GAA P10253 1/20 0.36
ALDH1A1 P00352 4/20 0.35
LMNA P02545 1/20 0.34
RAB9A P51151 1/20 0.34
GPR142 Q7Z601 1/20 0.33
NPC1 O15118 1/20 0.33
KMT2A Q03164 2/20 0.33
MEN1 O00255 1/20 0.33
ESR1 P03372 1/20 0.33
POLB P06746 1/20 0.33
MAPT P10636 1/20 0.33
BLM P54132 1/20 0.33
NPSR1 Q6W5P4 1/20 0.33
KLKB1 P03952 1/20 0.32
KLK1 P06870 1/20 0.32
HDAC3 O15379 1/20 0.32
HDAC1 Q13547 1/20 0.32
HDAC6 Q9UBN7 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Trifluoroacetic Acid SCHEMBL6503592 0.89 KDM4E (0.37) KDM4EGAAALDH1A1GPR142NPC1
SCHEMBL6531507 0.89 PARP1 (0.36) KDM4EGAAALDH1A1LMNARAB9A
SCHEMBL6505045 0.88 SMN1; SMN2 (0.35) KDM4EALDH1A1RAB9ANPC1KMT2A
SCHEMBL6504395 0.86 PPARA (0.37) GAAMAPTKLKB1
SCHEMBL6505593 0.86 ADORA2A (0.35) KDM4EALDH1A1RAB9ANPC1POLB
SCHEMBL6494741 0.85 PPARA (0.39) GAAKMT2AMEN1POLBMAPT
SCHEMBL6499174 0.85 ADORA1 (0.38) KDM4EGAAALDH1A1LMNARAB9A
SCHEMBL6495822 0.84 SHMT1 (0.39) KDM4EKMT2AMAPTKLKB1
SCHEMBL6498709 0.83 CDK2 (0.34) NPC1MAPTKLKB1
Trifluoroacetic Acid SCHEMBL6531504 0.79 PPARA (0.40) MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6884821-B1 Carboxylic acid derivatives and drugs containing the same EISAI CO., LTD. (JP) 2005-04-26 US disclosed
EP-1216980-A1 CARBOXYLIC ACID DERIVATIVES AND DRUGS CONTAINING THE SAME Eisai Co., Ltd. (JP) 2002-06-26 EP disclosed